Compile Data Set for Download or QSAR
Report error Found 209 Enz. Inhib. hit(s) with all data for entry = 1497
TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327284(N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)thio]-pheny...)
Affinity DataIC50: 10nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327241(N-[5-chloro-2-(methylsulfinyl)phenyl]-1-benzofuran...)
Affinity DataIC50: 11nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327214(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-3-(...)
Affinity DataIC50: 14nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327296(N-(2-{[(6-aminopyridin-2-yl)methyl]sulfonyl}-5-chl...)
Affinity DataIC50: 15nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327306(N-{5-chloro-2-[(1H-pyrazol-3-ylmethyl)thio]phenyl}...)
Affinity DataIC50: 16nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327377(N-{5-chloro-2-[(trifluoromethyl)sulfinyl]phenyl}-1...)
Affinity DataIC50: 19nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327325(N-{5-chloro-2-[(pyridin-3-ylmethyl)thio]phenyl}-1-...)
Affinity DataIC50: 22nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327385(N-{2-[(3-aminobenzyl)sulfonyl]-5-fluorophenyl}-1-b...)
Affinity DataIC50: 22nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327351(N-{2-[(3-aminobenzyl)sulfonyl]-5-chlorophenyl}-1-b...)
Affinity DataIC50: 23nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327268(4-chloro-N-[5-chloro-2-(methylthio)phenyl]-2-fluor...)
Affinity DataIC50: 25nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327332(N-(2-{[(5-amino-1H-pyrazol-3-yl)methyl]thio}-5-chl...)
Affinity DataIC50: 25nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327240(N-[5-chloro-2-(methylthio)phenyl]-1-benzofuran-2-s...)
Affinity DataIC50: 26nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327379(N-[2-(benzylsulfinyl)-5-chlorophenyl]-1-benzofuran...)
Affinity DataIC50: 27nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327295(N-(2-{[(6-aminopyridin-2-yl)methyl]sulfinyl}-5-chl...)
Affinity DataIC50: 28nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327338(N-{5-chloro-2-[(pyridin-2-ylmethyl)sulfinyl]-pheny...)
Affinity DataIC50: 29nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327339(N-{5-chloro-2-[(pyridin-2-ylmethyl)sulfonyl]-pheny...)
Affinity DataIC50: 29nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327294(N-(2-{[(6-aminopyridin-2-yl)methyl]thio}-5-chlorop...)
Affinity DataIC50: 32nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327328(N-{5-chloro-2-[(pyridin-3-ylmethyl)sulfonyl]-pheny...)
Affinity DataIC50: 32nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327357(N-(2-{[(5-amino-4H-1,2,4-triazol-3-yl)methyl]thio}...)
Affinity DataIC50: 32nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327380(N-[2-(benzylsulfonyl)-5-chlorophenyl]-1-benzofuran...)
Affinity DataIC50: 34nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327324(N-{5-chloro-2-[(pyridin-2-ylmethyl)thio]phenyl}-1-...)
Affinity DataIC50: 35nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327383(N-{2-[(3-aminobenzyl)sulfinyl]-5-fluorophenyl}-1-b...)
Affinity DataIC50: 38nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327350(N-{2-[(3-aminobenzyl)sulfinyl]-5-chlorophenyl}-1-b...)
Affinity DataIC50: 39nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327394(N-{2-[(3-aminobenzyl)sulfonyl]phenyl}-1-benzofuran...)
Affinity DataIC50: 41nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327242(N-[5-chloro-2-(methylsulfonyl)phenyl]-1-benzofuran...)
Affinity DataIC50: 42nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327320(N-(2-{[(2-amino-1,3-thiazol-4-yl)methyl]thio}-5-ch...)
Affinity DataIC50: 42nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327349(N-{2-[(3-aminobenzyl)thio]-5-chlorophenyl}-1-benzo...)
Affinity DataIC50: 42nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327232(3,4-dichloro-N-[5-chloro-2-(methylsulfinyl)phenyl]...)
Affinity DataIC50: 44nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327250(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-3-m...)
Affinity DataIC50: 44nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327238(4-chloro-N-[5-chloro-2-(ethylsulfinyl)phenyl]-3-(t...)
Affinity DataIC50: 50nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327421(N-[2-(benzylsulfinyl)-5-cyanophenyl]-1-benzofuran-...)
Affinity DataIC50: 50nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327280(4-chloro-N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)su...)
Affinity DataIC50: 51nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327261(N-[5-chloro-2-(methylsulfinyl)phenyl]-3-nitro-4-(t...)
Affinity DataIC50: 54nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327381(N-{2-[(3-aminobenzyl)thio]-5-fluorophenyl}-1-benzo...)
Affinity DataIC50: 55nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327354(N-{5-chloro-2-[(3-hydroxybenzyl)sulfonyl]phenyl}-1...)
Affinity DataIC50: 56nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327422(N-[2-(benzylsulfonyl)-5-cyanophenyl]-1-benzofuran-...)
Affinity DataIC50: 56nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327390(N-{2-[(3-aminobenzyl)sulfinyl]phenyl}-1-benzofuran...)
Affinity DataIC50: 58nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327281(N-{5-chloro-2-[(1H-imidazol-2-ylmethyl)thio]-pheny...)
Affinity DataIC50: 60nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327271(3-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-2-f...)
Affinity DataIC50: 61nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327248(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]benz...)
Affinity DataIC50: 62nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327215(4-chloro-N-[5-chloro-2-(methylsulfonyl)phenyl]-3-(...)
Affinity DataIC50: 64nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327278(4-chloro-N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)th...)
Affinity DataIC50: 68nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327262(N-[5-chloro-2-(methylthio)phenyl]-5-methylfuran-2-...)
Affinity DataIC50: 70nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327376(N-{5-chloro-2-[(trifluoromethyl)sulfonyl]phenyl}-1...)
Affinity DataIC50: 73nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327399(N-{5-chloro-2-[(2-nitrobenzyl)sulfinyl]phenyl}-1-b...)
Affinity DataIC50: 75nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327236(4-chloro-N-{5-chloro-2-[(3-hydroxycyclopentyl)sulf...)
Affinity DataIC50: 76nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
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TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327289(3-({2-[(1-benzofuran-2-ylsulfonyl)amino]-4-chlorop...)
Affinity DataIC50: 76nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327326(N-{5-chloro-2-[(pyridin-3-ylmethyl)sulfinyl]phenyl...)
Affinity DataIC50: 76nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327352(N-{5-chloro-2-[(3-hydroxybenzyl)thio]phenyl}-1-ben...)
Affinity DataIC50: 77nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
Go to US Patent

TargetC-C chemokine receptor type 2(Human)
Allergan

US Patent
LigandPNGBDBM327373(N-(5-chloro-2-{[(2-fluoropyridin-3-yl)methyl]-sulf...)
Affinity DataIC50: 79nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
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