Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 8160
LigandPNGBDBM235633(US9388170, 20)
Affinity DataIC50: 6.80nMAssay Description:BT474 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
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LigandPNGBDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50: 47nMAssay Description:BT474 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
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PDB3D3D Structure (crystal)
LigandPNGBDBM50123190(CHEMBL3622645 | US9388170, 13)
Affinity DataIC50: 57nMAssay Description:BT474 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
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LigandPNGBDBM235633(US9388170, 20)
Affinity DataIC50: 100nMAssay Description:BT474 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
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LigandPNGBDBM50123190(CHEMBL3622645 | US9388170, 13)
Affinity DataIC50: 100nMAssay Description:BT474 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
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LigandPNGBDBM235633(US9388170, 20)
Affinity DataIC50: 1.79E+3nMAssay Description:A431 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 100...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
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LigandPNGBDBM50123190(CHEMBL3622645 | US9388170, 13)
Affinity DataIC50: 3.10E+3nMAssay Description:A431 Cell Line: 1. 5×103 cells per well in 100 μl of medium were seeded in 96-well plate, here the medium contained 5% FBS2. 24 hours later, 100...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details
Go to US Patent