Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 12090
TargetProlyl endopeptidase FAP(Human)
Nuclidium

US Patent
LigandPNGBDBM677071(US20240173440, Compound [natCu]Cu-NODAGA-F3)
Affinity DataIC50: 0.0400nMAssay Description:The enzymatic activity of hFAP on the substrate Z-Gly-Pro-AMC was measured at room temperature on a microtiter plate reader, monitoring the fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2024
Entry Details
Go to US Patent

TargetProlyl endopeptidase FAP(Human)
Nuclidium

US Patent
LigandPNGBDBM677073(US20240173440, Compound [natCu]Cu-NODAGA-F4)
Affinity DataIC50: 0.105nMAssay Description:The enzymatic activity of hFAP on the substrate Z-Gly-Pro-AMC was measured at room temperature on a microtiter plate reader, monitoring the fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2024
Entry Details
Go to US Patent

TargetProlyl endopeptidase FAP(Human)
Nuclidium

US Patent
LigandPNGBDBM677072(US20240173440, Compound [natCu]Cu-NODAGA-F2)
Affinity DataIC50: 0.120nMAssay Description:The enzymatic activity of hFAP on the substrate Z-Gly-Pro-AMC was measured at room temperature on a microtiter plate reader, monitoring the fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2024
Entry Details
Go to US Patent

TargetProlyl endopeptidase FAP(Human)
Nuclidium

US Patent
LigandPNGBDBM677070(US20240173440, Compound [natCu]Cu- NODAGA-F1)
Affinity DataIC50: 0.141nMAssay Description:The enzymatic activity of hFAP on the substrate Z-Gly-Pro-AMC was measured at room temperature on a microtiter plate reader, monitoring the fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2024
Entry Details
Go to US Patent