Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 11335
TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608309(US11691981, Compound 66)
Affinity DataIC50: 4nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608284(US11691981, Compound 41)
Affinity DataIC50: 12nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608255(US11691981, Compound 17)
Affinity DataIC50: 12nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608288(US11691981, Compound 45)
Affinity DataIC50: 13nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608336(US11691981, Compound 73)
Affinity DataIC50: 14nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608308(US11691981, Compound 65)
Affinity DataIC50: 14nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM50564603(CHEMBL4777294 | US11691981, Compound 77)
Affinity DataIC50: 17nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608337(US11691981, Compound 74)
Affinity DataIC50: 17nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608281(US11691981, Compound 38)
Affinity DataIC50: 18nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608296(US11691981, Compound 53)
Affinity DataIC50: 18nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608271(US11691981, Compound 29)
Affinity DataIC50: 19nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608295(US11691981, Compound 52)
Affinity DataIC50: 21nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608300(US11691981, Compound 57)
Affinity DataIC50: 21nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM50564620(Ly-3200882 | Ly3200882 | US11691981, Compound A)
Affinity DataIC50: 22nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608341(US11691981, Compound 78)
Affinity DataIC50: 22nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608247(US11691981, Compound 11)
Affinity DataIC50: 24nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608314(US11691981, Compound 71)
Affinity DataIC50: 25nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608248(US11691981, Compound 12)
Affinity DataIC50: 28nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608342(US11691981, Compound 79)
Affinity DataIC50: 29nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608305(US11691981, Compound 62)
Affinity DataIC50: 29nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608307(US11691981, Compound 64)
Affinity DataIC50: 32nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608302(US11691981, Compound 59)
Affinity DataIC50: 32nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608292(US11691981, Compound 49)
Affinity DataIC50: 32nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608254(US11691981, Compound 16)
Affinity DataIC50: 34nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608298(US11691981, Compound 55)
Affinity DataIC50: 35nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608269(US11691981, Compound 28)
Affinity DataIC50: 35nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608250(US11691981, Compound 14)
Affinity DataIC50: 37nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608261(US11691981, Compound 21)
Affinity DataIC50: 37nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608263(US11691981, Compound 23)
Affinity DataIC50: 38nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608301(US11691981, Compound 58)
Affinity DataIC50: 39nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608277(US11691981, Compound 34)
Affinity DataIC50: 42nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608239(US11691981, Compound 5)
Affinity DataIC50: 43nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608249(US11691981, Compound 13)
Affinity DataIC50: 44nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608240(US11691981, Compound 6)
Affinity DataIC50: 46nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608260(US11691981, Compound 20)
Affinity DataIC50: 48nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608276(US11691981, Compound 33)
Affinity DataIC50: 49nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608303(US11691981, Compound 60)
Affinity DataIC50: 50nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608310(US11691981, Compound 67)
Affinity DataIC50: 51nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608343(US11691981, Compound 80 | US11691981, Compound 81)
Affinity DataIC50: 51nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608235(US11691981, Compound 2)
Affinity DataIC50: 53nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608262(US11691981, Compound 22)
Affinity DataIC50: 54nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608294(US11691981, Compound 51)
Affinity DataIC50: 55nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608279(US11691981, Compound 36)
Affinity DataIC50: 56nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608297(US11691981, Compound 54)
Affinity DataIC50: 56nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608343(US11691981, Compound 80 | US11691981, Compound 81)
Affinity DataIC50: 57nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608241(US11691981, Compound 7 | US11691981, Compound 27)
Affinity DataIC50: 58nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608238(US11691981, Compound 4)
Affinity DataIC50: 60nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608234(US11691981, Compound 1)
Affinity DataIC50: 61nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608289(US11691981, Compound 46)
Affinity DataIC50: 66nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608265(US11691981, Compound 25)
Affinity DataIC50: 66nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent

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