Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 11251
TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602767(US11649233, Compound 34 | Synthesis of (Z)-6-((2-(...)
Affinity DataIC50: 6nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602764(US11649233, Compound 31 | Synthesis of (Z)-5-((2-(...)
Affinity DataIC50: 11nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602765(US11649233, Compound 32 | Synthesis of (Z)-6-((2-(...)
Affinity DataIC50: 11nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602761(US11649233, Compound 28 | Synthesis of (Z)-3-((2-(...)
Affinity DataIC50: 14nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602756(US11649233, Compound 23 | Synthesis of (Z)-2-((2-(...)
Affinity DataIC50: 14nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602766(US11649233, Compound 33)
Affinity DataIC50: 14nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602760(US11649233, Compound 27 | Synthesis of (E)-3-((2-(...)
Affinity DataIC50: 16nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602750(US11649233, Compound 5 | Synthesis of (E)-6-((2-(a...)
Affinity DataIC50: 18nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602755(US11649233, Compound 21 | Synthesis of (E)-6-((2-(...)
Affinity DataIC50: 21nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602754(US11649233, Compound 19 | Synthesis of (E)-5-((2-(...)
Affinity DataIC50: 21nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602752(US11649233, Compound 16 | Synthesis of (E)-5-((2-(...)
Affinity DataIC50: 24nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602757(US11649233, Compound 24 | Synthesis of (E)-2-((2-(...)
Affinity DataIC50: 24nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602762(US11649233, Compound 29 | Synthesis of (Z)-5-((2-(...)
Affinity DataIC50: 25nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602758(US11649233, Compound 25 | Synthesis of (Z)-2-((2-(...)
Affinity DataIC50: 25nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602751(US11649233, Compound 8 | Synthesis of (E)-3-((2-(a...)
Affinity DataIC50: 30nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602763(US11649233, Compound 30 | Synthesis of (E)-5-((2-(...)
Affinity DataIC50: 32nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602759(US11649233, Compound 26 | Synthesis of (E)-2-((2-(...)
Affinity DataIC50: 51nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [copper-containing] 3(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602749(US11649233, Compound 4 | Synthesis of (E)-6-((2-(a...)
Affinity DataIC50: 59nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [flavin-containing] B(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602750(US11649233, Compound 5 | Synthesis of (E)-6-((2-(a...)
Affinity DataIC50: 1.30E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602752(US11649233, Compound 16 | Synthesis of (E)-5-((2-(...)
Affinity DataIC50: 2.80E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602762(US11649233, Compound 29 | Synthesis of (Z)-5-((2-(...)
Affinity DataIC50: 4.10E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602763(US11649233, Compound 30 | Synthesis of (E)-5-((2-(...)
Affinity DataIC50: 5.80E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602750(US11649233, Compound 5 | Synthesis of (E)-6-((2-(a...)
Affinity DataIC50: 6.30E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602765(US11649233, Compound 32 | Synthesis of (Z)-6-((2-(...)
Affinity DataIC50: 6.60E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602767(US11649233, Compound 34 | Synthesis of (Z)-6-((2-(...)
Affinity DataIC50: 8.40E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
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TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602766(US11649233, Compound 33)
Affinity DataIC50: 8.60E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602759(US11649233, Compound 26 | Synthesis of (E)-2-((2-(...)
Affinity DataIC50: 8.80E+3nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] B(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602756(US11649233, Compound 23 | Synthesis of (Z)-2-((2-(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602758(US11649233, Compound 25 | Synthesis of (Z)-2-((2-(...)
Affinity DataIC50: 1.30E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602755(US11649233, Compound 21 | Synthesis of (E)-6-((2-(...)
Affinity DataIC50: 1.40E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602756(US11649233, Compound 23 | Synthesis of (Z)-2-((2-(...)
Affinity DataIC50: 1.90E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602761(US11649233, Compound 28 | Synthesis of (Z)-3-((2-(...)
Affinity DataIC50: 2.00E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602757(US11649233, Compound 24 | Synthesis of (E)-2-((2-(...)
Affinity DataIC50: 3.70E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602760(US11649233, Compound 27 | Synthesis of (E)-3-((2-(...)
Affinity DataIC50: 3.80E+4nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] B(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602755(US11649233, Compound 21 | Synthesis of (E)-6-((2-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
Nanjing Transthera Biosciences

US Patent
LigandPNGBDBM602751(US11649233, Compound 8 | Synthesis of (E)-3-((2-(a...)
Affinity DataIC50: 1.00E+5nMAssay Description:Test substances: the compounds of the present invention shown in Table 1 and prepared according to the methods of the examples 1. Inhibition Activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
Go to US Patent