Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 10732
LigandPNGBDBM562408(US11401279, Example 2)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468549(4-((2-(2,2'- dichloro- 3'-(5- isopropyl-1- methyl-...)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468552(4-((2-(2,2′-dichloro-3′-(5-(2-hydroxye...)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562433(US11401279, Example 66)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562425(US11401279, Example 51)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562424(US11401279, Example 49)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562420(US11401279, Example 15)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562419(US11401279, Example 12)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562417(US11401279, Example 11)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562415(US11401279, Example 8)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562410(US11401279, Example 3)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562416(US11401279, Example 10)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562412(US11401279, Example 7)
Affinity DataIC50: 1.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468553((S)-4- ((2-(2,2'- dichloro- 3'-(5-(2- hydroxy- pro...)
Affinity DataIC50: 1.60nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562421(US11401279, Example 16)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562422(US11401279, Example 47)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562409(US11401279, Example 9)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468553((S)-4- ((2-(2,2'- dichloro- 3'-(5-(2- hydroxy- pro...)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562413(US11401279, Example 14)
Affinity DataIC50: 1.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562429(US11401279, Example 56)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562432(US11401279, Example 65)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562445(US11401279, Example 183)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562418(US11401279, Example 13)
Affinity DataIC50: 1.80nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562411(US11401279, Example 4)
Affinity DataIC50: 1.90nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468550(4-((2-(2,2'- dichloro- 3'-(5- cyclobutyl-1- methyl...)
Affinity DataIC50: 1.90nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562423(US11401279, Example 48)
Affinity DataIC50: 2nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562428(US11401279, Example 55)
Affinity DataIC50: 2.10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562414(US11401279, Example 5)
Affinity DataIC50: 2.10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562430(US11401279, Example 61)
Affinity DataIC50: 2.20nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562407(US11401279, Example 1)
Affinity DataIC50: 2.20nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM395657(US10308644, Example 267 | (R)-4-((2-(2-chloro-3...)
Affinity DataIC50: 2.30nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM395655(US10308644, Example 265 | (R)-4-(2-(2-(2- chloro-3...)
Affinity DataIC50: 2.30nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468460(US10806785, Example 102 | 4-((2-((2'- chloro-3'-(1...)
Affinity DataIC50: 2.40nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562434(US11401279, Example 69)
Affinity DataIC50: 2.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562431(US11401279, Example 63)
Affinity DataIC50: 2.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562427(US11401279, Example 53)
Affinity DataIC50: 2.5nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM562426(US11401279, Example 52)
Affinity DataIC50: 2.70nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468548(4-((2-(2,2′-dichloro-3′-(5-ethyl-1-met...)
Affinity DataIC50: 2.90nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468479(4-((2-((2- chloro-3'-(1,5- dimethyl-4,5,6,7- tetra...)
Affinity DataIC50: 3.40nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468442(US10806785, Example 84 | 4-((2-((2,2′-dichlo...)
Affinity DataIC50: 8.30nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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Date in BDB:
10/23/2022
Entry Details
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LigandPNGBDBM468551(4-((2-(2,2'- dichloro- 3'-(1- methyl-5- (tetrahydr...)
Affinity DataIC50: 18nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
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Date in BDB:
10/23/2022
Entry Details
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