Compile Data Set for Download or QSAR
Report error Found 137 Enz. Inhib. hit(s) with all data for entry = 8923
TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429526(3-(5-Chloro-6-isobutoxypyridin-3-yl)-N-(cyclopropy...)
Affinity DataIC50: 3.40nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429525(3-(5-Chloro-6-isobutoxypyridin-3-yl)-5-fluoro-1-me...)
Affinity DataIC50: 11nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465061(CHEMBL4290933 | US10550080, Example 47)
Affinity DataIC50: 16nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429496(3-(5-Chloro-6-isobutoxypyridin-3-yl)-N-(cyclopropy...)
Affinity DataIC50: 22nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465063(CHEMBL4287506 | US10550080, Example 45)
Affinity DataIC50: 26nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465064(CHEMBL4294322 | US10550080, Example 36)
Affinity DataIC50: 38nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465060(CHEMBL4276864 | US10550080, Example 49)
Affinity DataIC50: 38nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465061(CHEMBL4290933 | US10550080, Example 47)
Affinity DataIC50: 39nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465057(CHEMBL4292013 | US10550080, Example 46)
Affinity DataIC50: 49nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465059(CHEMBL4283748 | US10550080, Example 35)
Affinity DataIC50: 52nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465063(CHEMBL4287506 | US10550080, Example 45)
Affinity DataIC50: 59nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465058(CHEMBL4280298 | US10550080, Example 39)
Affinity DataIC50: 66nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465058(CHEMBL4280298 | US10550080, Example 39)
Affinity DataIC50: 67nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429511(N-(cyclopropylsulfonyl)-3-(4-(difluoromethyl)pheny...)
Affinity DataIC50: 69nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429490(N-(cyclopropylsulfonyl)-1-methyl-3-(4-(trifluorome...)
Affinity DataIC50: 77nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429470(1-Methyl-N-(methylsulfonyl)-3-(4-(trifluoromethoxy...)
Affinity DataIC50: 80nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465057(CHEMBL4292013 | US10550080, Example 46)
Affinity DataIC50: 84nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429453(1-Methyl-N-(methylsulfonyl)-3-(4-(trifluoromethyl)...)
Affinity DataIC50: 85nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465059(CHEMBL4283748 | US10550080, Example 35)
Affinity DataIC50: 86nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429527(5-Fluoro-3-(6-isobutoxypyridin-3-yl)-1-methyl-N-(m...)
Affinity DataIC50: 86nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429509(3-(5-Chloro-6-isobutoxypyridin-3-yl)-1-isopropyl-N...)
Affinity DataIC50: 89nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465062(CHEMBL4279180 | US10550080, Example 2)
Affinity DataIC50: 90nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465062(CHEMBL4279180 | US10550080, Example 2)
Affinity DataIC50: 91nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429532(3-(4-(Difluoromethyl)phenyl)-5-fluoro-1-methyl-N-(...)
Affinity DataIC50: 91nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429527(5-Fluoro-3-(6-isobutoxypyridin-3-yl)-1-methyl-N-(m...)
Affinity DataIC50: 104nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429490(N-(cyclopropylsulfonyl)-1-methyl-3-(4-(trifluorome...)
Affinity DataIC50: 109nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465060(CHEMBL4276864 | US10550080, Example 49)
Affinity DataIC50: 146nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50465064(CHEMBL4294322 | US10550080, Example 36)
Affinity DataIC50: 154nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429519(N-(tert-butylsulfonyl)-3-(5-chloro-6-isobutoxypyri...)
Affinity DataIC50: 156nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429486(3-(4-Ethylphenyl)-1-methyl-N-(methylsulfonyl)-1H-i...)
Affinity DataIC50: 173nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429495(3-(6-Isobutoxypyridin-3-yl)-1-methyl-N-(methylsulf...)
Affinity DataIC50: 183nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429514(3-(5-Chloro-6-(cyclopropylmethoxy)pyridin-3-yl)-1-...)
Affinity DataIC50: 189nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429523(3-(5-Chloro-6-isobutoxypyridin-3-yl)-N-(cyclopropy...)
Affinity DataIC50: 195nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429517(3-(5-Chloro-6-isobutoxypyridin-3-yl)-N-(isopropyls...)
Affinity DataIC50: 207nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429488(3-(3-Isopropylphenyl)-1-methyl-N-(methylsulfonyl)-...)
Affinity DataIC50: 217nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429489(3-(3-Ethylphenyl)-1-methyl-N-(methylsulfonyl)-1H-i...)
Affinity DataIC50: 220nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429470(1-Methyl-N-(methylsulfonyl)-3-(4-(trifluoromethoxy...)
Affinity DataIC50: 243nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429510(3-(4-(Difluoromethyl)phenyl)-1-methyl-N-(methylsul...)
Affinity DataIC50: 262nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429514(3-(5-Chloro-6-(cyclopropylmethoxy)pyridin-3-yl)-1-...)
Affinity DataIC50: 270nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429494(3-(4-Isobutoxyphenyl)-1-methyl-N-(methylsulfonyl)-...)
Affinity DataIC50: 275nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429484(1-Methyl-N-(methylsulfonyl)-3-(3-(trifluoromethyl)...)
Affinity DataIC50: 290nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429496(3-(5-Chloro-6-isobutoxypyridin-3-yl)-N-(cyclopropy...)
Affinity DataIC50: 294nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429526(3-(5-Chloro-6-isobutoxypyridin-3-yl)-N-(cyclopropy...)
Affinity DataIC50: 310nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429482(3-(4-Isobutylphenyl)-1-methyl-N-(methylsulfonyl)-1...)
Affinity DataIC50: 317nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429511(N-(cyclopropylsulfonyl)-3-(4-(difluoromethyl)pheny...)
Affinity DataIC50: 321nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429492(1-Methyl-N-(thiophen-2-ylsulfonyl)-3-(4-(trifluoro...)
Affinity DataIC50: 361nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429482(3-(4-Isobutylphenyl)-1-methyl-N-(methylsulfonyl)-1...)
Affinity DataIC50: 363nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429487(1-Methyl-N-(methylsulfonyl)-3-(m-tolyl)-1H-indole-...)
Affinity DataIC50: 375nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429492(1-Methyl-N-(thiophen-2-ylsulfonyl)-3-(4-(trifluoro...)
Affinity DataIC50: 419nMAssay Description:Ion Works Barracuda population patch clamp (PPC). PPC measurements were performed using an IonWorks Barracuda instrument (Molecular Devices Corporati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
Go to US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM429453(1-Methyl-N-(methylsulfonyl)-3-(4-(trifluoromethyl)...)
Affinity DataIC50: 422nMAssay Description:hNaV1.7 binding affinities were determined with a filtration binding assay using purified membranes from HEK293 cells stably expressing hNaV1.7. HEK2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
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