Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 8703
TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413601(US10421722, Compound 9b)
Affinity DataKi:  2.30nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413594(US10421722, Compound 3)
Affinity DataKi:  2.40nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413600(US10421722, Compound 9a)
Affinity DataKi:  2.40nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM70577(US10421722, Compound 2)
Affinity DataKi:  5.40nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413597(US10421722, Compound 6a)
Affinity DataKi:  6.30nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413596(US10421722, Compound 4)
Affinity DataKi:  6.5nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM50018078(CHEMBL20943 | V-100 | 2-(4-Phenyl-piperidin-1-yl)-...)
Affinity DataKi:  9.90nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413599(US10421722, Compound 7)
Affinity DataKi:  12.8nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
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TargetVesicular acetylcholine transporter(Human)
Washington University

US Patent
LigandPNGBDBM413598(US10421722, Compound 6b)
Affinity DataKi:  13nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2020
Entry Details
Go to US Patent