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Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 3013
TargetSodium/glucose cotransporter 2(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM254941(US9505734, I-D1-6 | US10294259, Compound Table 3.2)
Affinity DataIC50: 0.670nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM388440(US10294259, Compound Table 3.1)
Affinity DataIC50: 3.30nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM388442(US10294259, Compound Table 3.3)
Affinity DataIC50: 7.80nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM388440(US10294259, Compound Table 3.1)
Affinity DataIC50: 86nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM388442(US10294259, Compound Table 3.3)
Affinity DataIC50: 187nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM254941(US9505734, I-D1-6 | US10294259, Compound Table 3.2)
Affinity DataIC50: 251nMAssay Description:IC50 values of inhibition of some compounds described in the present invention and related compounds on SGLT2 and SGLT1 are determined according to t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2020
Entry Details
Go to US Patent