Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 2474
TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM367610(US10227310, Example 2 | N-[(1S)-2-[4-[2- (4-Amino-...)
Affinity DataIC50: 54.4nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
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TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM367613(US10227310, Example 66 | N-[(1S)-2-[4-[2-(4-Amino-...)
Affinity DataIC50: 68.9nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
Go to US Patent

TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM367612(US10227310, Example 42 | N-[(1S)-2-[4-[2-(4-Amino-...)
Affinity DataIC50: 96.4nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
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TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM367615(US10227310, Example 71 | Methyl N-[(1S)-2-[4-[2-(4...)
Affinity DataIC50: 149nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
Go to US Patent

TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM367614(US10227310, Example 69 | N-[(1S)-2-[4-[2-(4-Amino-...)
Affinity DataIC50: 170nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
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TargetGhrelin O-acyltransferase(Human)
Eli Lilly

US Patent
LigandPNGBDBM367611(US10227310, Example 37 | N-[(1S)-2-[(4R,S)- 4-[2-(...)
Affinity DataIC50: 574nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
Go to US Patent