Compile Data Set for Download or QSAR
Report error Found 113 Enz. Inhib. hit(s) with all data for entry = 50005757
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040583((R)-4-(1,3-Dioxo-5-propoxy-1,3-dihydro-isoindol-2-...)
Affinity DataIC50: 2.10nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040607((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 3.80nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040600((R)-4-(1,3-Dioxo-5-phenyl-1,3-dihydro-isoindol-2-y...)
Affinity DataIC50: 4.5nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040585((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50: 4.80nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040593((R)-4-(5,7-Dioxo-5,7-dihydro-[1,3]dioxolo[4,5-f]is...)
Affinity DataIC50: 5nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 5nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040610((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 6.70nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040597((R)-4-(4-Methoxy-1,3-dioxo-1,3-dihydro-benzo[f]iso...)
Affinity DataIC50: 7.40nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040596((R)-4-(1,3-Dioxo-1,3-dihydro-pyrrolo[3,4-b]quinoli...)
Affinity DataIC50: 7.5nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040616((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 11nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040592((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 12nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040593((R)-4-(5,7-Dioxo-5,7-dihydro-[1,3]dioxolo[4,5-f]is...)
Affinity DataIC50: 12nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040609((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 13nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040613((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 14nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040579((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 15nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040614((R)-4-(5-Methoxy-1,3-dioxo-1,3-dihydro-benzo[f]iso...)
Affinity DataIC50: 15nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040583((R)-4-(1,3-Dioxo-5-propoxy-1,3-dihydro-isoindol-2-...)
Affinity DataIC50: 15nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040600((R)-4-(1,3-Dioxo-5-phenyl-1,3-dihydro-isoindol-2-y...)
Affinity DataIC50: 19nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040613((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 19nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 20nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040596((R)-4-(1,3-Dioxo-1,3-dihydro-pyrrolo[3,4-b]quinoli...)
Affinity DataIC50: 22nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040580((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 27nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040605((R)-4-(6-Bromo-1,3-dioxo-1H,3H-benzo[de]isoquinoli...)
Affinity DataIC50: 28nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040607((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 29nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040595((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 30nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040611((R)-2-((S)-1-Benzylcarbamoyl-3-methyl-butylamino)-...)
Affinity DataIC50: 32nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040589((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 35nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040602((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 36nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040615((R)-4-(6-Methoxy-1,3-dioxo-1,3-dihydro-benzo[f]iso...)
Affinity DataIC50: 36nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040614((R)-4-(5-Methoxy-1,3-dioxo-1,3-dihydro-benzo[f]iso...)
Affinity DataIC50: 36nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040590((R)-2-[(S)-1-(Benzyl-methyl-carbamoyl)-3-methyl-bu...)
Affinity DataIC50: 37nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040585((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50: 38nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040579((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 41nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040609((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 44nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040601((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50: 49nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040616((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 49nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040592((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 51nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040603((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 54nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040597((R)-4-(4-Methoxy-1,3-dioxo-1,3-dihydro-benzo[f]iso...)
Affinity DataIC50: 54nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040599(4-({(S)-2-[(R)-1-Carboxy-3-(1,3-dioxo-1,3-dihydro-...)
Affinity DataIC50: 56nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040590((R)-2-[(S)-1-(Benzyl-methyl-carbamoyl)-3-methyl-bu...)
Affinity DataIC50: 57nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040582((R)-4-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-2-[(S)...)
Affinity DataIC50: 59nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040586((R)-2-[(S)-3-Methyl-1-((S)-1-methylcarbamoyl-2-phe...)
Affinity DataIC50: 63nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040591((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 69nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040587((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 70nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040603((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 70nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040610((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 70nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040607((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 72nMAssay Description:Activity against human stromelysin (MMP-3).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040599(4-({(S)-2-[(R)-1-Carboxy-3-(1,3-dioxo-1,3-dihydro-...)
Affinity DataIC50: 74nMAssay Description:Activity against human gelatinase (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Glaxo Inc. Research Institute

Curated by ChEMBL
LigandPNGBDBM50040606((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50: 74nMAssay Description:Activity against human collagenase (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 113 total ) | Next | Last >>
Jump to: