Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50012249
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50555899(CHEMBL1683636)
Affinity DataIC50: 60nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50053584(CHEMBL1977874)
Affinity DataIC50: 280nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50555900(CHEMBL4776943)
Affinity DataIC50: 310nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50126829((E)-1-(6-(3-acetyl-2,4,6-trihydroxy-5-methylbenzyl...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50555901(CHEMBL4516025)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of eEF2K (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed