Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50009309
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527005(CHEMBL15908)
Affinity DataEC50: >6.00E+3nMAssay Description:Agonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50266165((S)-N-(2-oxotetrahydrofuran-3-yl)-2-(4-(trifluorom...)
Affinity DataEC50:  1.40E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  139nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50241433((S)-3-(4-bromophenyl)-N-(2-oxotetrahydrofuran-3-yl...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527017(CHEMBL4461584)
Affinity DataEC50:  71nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527002(CHEMBL4444462)
Affinity DataEC50:  1.70E+4nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527018(CHEMBL4517457)
Affinity DataEC50:  250nMAssay Description:Agonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527003(CHEMBL4522587)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527004(CHEMBL4450449)
Affinity DataEC50:  4.20E+3nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526984(CHEMBL4579576)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50351511(CHEMBL463321)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526977(CHEMBL4462112)
Affinity DataEC50:  2.60E+3nMAssay Description:Activation of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526983(CHEMBL4535946)
Affinity DataEC50:  500nMAssay Description:Agonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527015(CHEMBL4527540)
Affinity DataIC50: 130nMAssay Description:Inhibition of Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50266165((S)-N-(2-oxotetrahydrofuran-3-yl)-2-(4-(trifluorom...)
Affinity DataIC50: 600nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50266163((S)-2-(4-iodophenyl)-N-(2-oxotetrahydrofuran-3-yl)...)
Affinity DataIC50: 900nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50266164((S)-2-(4-nitrophenyl)-N-(2-oxotetrahydrofuran-3-yl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50373105(CHEMBL259441)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50300132(N-heptanoyl-L-homoserine lactone | CHEMBL584972)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527006(CHEMBL16191)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527019(CHEMBL15876)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50373048(CHEMBL184106)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526979(CHEMBL16015)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527014(CHEMBL16014)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526985(CHEMBL15678)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50351251(CHEMBL1818523)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526978(CHEMBL273574)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50266165((S)-N-(2-oxotetrahydrofuran-3-yl)-2-(4-(trifluorom...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526986(CHEMBL15893)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527016(CHEMBL184464)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50300131(N-(4-bromophenylacetanoyl)-L-homoserine lactone | ...)
Affinity DataIC50: 3.70E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526987(CHEMBL15975)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526990(CHEMBL277954)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526988(CHEMBL15125)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527012(CHEMBL4571277)
Affinity DataIC50: 4.10E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527001(CHEMBL1823942)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50351511(CHEMBL463321)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527007(CHEMBL16100)
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526996(CHEMBL4284234)
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR transfected with lasB-GFP by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527009(CHEMBL426064)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526993(CHEMBL184178)
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526982(CHEMBL4549418)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526994(CHEMBL184703)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526989(CHEMBL15839)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50241433((S)-3-(4-bromophenyl)-N-(2-oxotetrahydrofuran-3-yl...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526992(CHEMBL359766)
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527020(CHEMBL4538227)
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at LasR in Pseudomonas aeruginosa harboring plasI-LVAgfp assessed as inhibition of GFP production incubated for 6 hrs by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526995(CHEMBL184295)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50526976(CHEMBL1615001)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Larkin University

Curated by ChEMBL
LigandPNGBDBM50527010(CHEMBL4434909)
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 65 total ) | Next | Last >>
Jump to: