Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50010437
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataKd:  3.10nMAssay Description:Binding affinity to GAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538885(CHEMBL4646895)
Affinity DataIC50: 22nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538901(CHEMBL4642467)
Affinity DataIC50: 24nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50288800(CHEMBL4172550)
Affinity DataIC50: 39nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538879(CHEMBL4645917)
Affinity DataIC50: 42nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538876(CHEMBL4642620)
Affinity DataIC50: 71nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538890(CHEMBL4636314)
Affinity DataIC50: 73nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538887(CHEMBL4643096)
Affinity DataIC50: 83nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538900(CHEMBL4641825)
Affinity DataIC50: 99nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538888(CHEMBL4632903)
Affinity DataIC50: 101nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538897(CHEMBL4639991)
Affinity DataIC50: 110nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538891(CHEMBL4638602)
Affinity DataIC50: 113nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538886(CHEMBL4632372)
Affinity DataIC50: 118nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538904(CHEMBL4633404)
Affinity DataIC50: 124nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538905(CHEMBL4642058)
Affinity DataIC50: 126nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538892(CHEMBL4640730)
Affinity DataIC50: 132nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50086277(CHEMBL3425876)
Affinity DataIC50: 136nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538903(CHEMBL4635935)
Affinity DataIC50: 136nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538893(CHEMBL4640641)
Affinity DataIC50: 173nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538899(CHEMBL4648802)
Affinity DataIC50: 214nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538898(CHEMBL4638387)
Affinity DataIC50: 262nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538895(CHEMBL4648554)
Affinity DataIC50: 364nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538889(CHEMBL4644472)
Affinity DataIC50: 370nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538894(CHEMBL4635431)
Affinity DataIC50: 370nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538896(CHEMBL4648514)
Affinity DataIC50: 370nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538902(CHEMBL4637058)
Affinity DataIC50: 422nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538883(CHEMBL4634338)
Affinity DataIC50: 458nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538877(CHEMBL4636735)
Affinity DataIC50: 545nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538875(CHEMBL4642436)
Affinity DataIC50: 661nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538882(CHEMBL4639109)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538881(CHEMBL4636582)
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538880(CHEMBL4638607)
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538878(CHEMBL4648166)
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCyclin-G-associated kinase(Human)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50538884(CHEMBL4642223)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed