Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50046792
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in human HEK293T cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]PK11195 from TSPO in human HEK293T cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  806nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed
TargetTranslocator protein(Human)
University of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2016
Entry Details Article
PubMed