Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50045178
TargetPhosphatidylinositol 3-kinase C2 domain-containing subunit gamma(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048418(CHEMBL3360227)
Affinity DataIC50: 340nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048419(CHEMBL3360231)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2beta assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 3-kinase C2 domain-containing subunit gamma(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048416(CHEMBL3360219)
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 3-kinase C2 domain-containing subunit gamma(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048417(CHEMBL3360221)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 3-kinase C2 domain-containing subunit gamma(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048419(CHEMBL3360231)
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048418(CHEMBL3360227)
Affinity DataIC50: 2.88E+4nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2beta assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048416(CHEMBL3360219)
Affinity DataIC50: 4.48E+4nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2beta assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Human)
Eberhard Karls University Tuebingen

Curated by ChEMBL
LigandPNGBDBM50048417(CHEMBL3360221)
Affinity DataIC50: 6.12E+4nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2beta assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed