Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50044414
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016496(CHEMBL3260241)
Affinity DataIC50: 30nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016508(CHEMBL3260249)
Affinity DataIC50: 90nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016502(CHEMBL3260248)
Affinity DataIC50: 120nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016495(CHEMBL3260236)
Affinity DataIC50: 190nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016501(CHEMBL3260247)
Affinity DataIC50: 190nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016498(CHEMBL3260243)
Affinity DataIC50: 590nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016500(CHEMBL3260246)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016497(CHEMBL3260242)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016499(CHEMBL3260244)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50016509(CHEMBL3260250)
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of PLK1 (unknown origin) using RRRDELMEASFADQEAKV as substrate after 20 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed