Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50043391
TargetCyclin-dependent kinase 5 activator 1(Human)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50077360(3,10-Dihydroxy-13-(3-hydroxy-4-methoxy-phenyl)-2,1...)
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50077360(3,10-Dihydroxy-13-(3-hydroxy-4-methoxy-phenyl)-2,1...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50077360(3,10-Dihydroxy-13-(3-hydroxy-4-methoxy-phenyl)-2,1...)
Affinity DataIC50: 55nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Mouse)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 150nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using RS peptide and [gamma-33P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 220nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 220nMAssay Description:Inhibition of PIM1 (unknown origin) expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 440nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 440nMAssay Description:Inhibition of human recombinant DYRK1A expressed in Escherichia coli using [gamma-33P]ATP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Mouse)
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50440393(CHEMBL2425487)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse recombinant CLK3 expressed in Escherichia coli using RS peptide and [gamma-33P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed