Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50040683
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50356012(AAPTAMINE)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398322(HETERONEMIN)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398323(CHEMBL508487)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398324(CHEMBL510804)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398325(CHEMBL2177350)
Affinity DataEC50:  8.70E+3nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398326(CHEMBL2177349)
Affinity DataEC50:  1.48E+4nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398327(VARIOLIN B)
Affinity DataEC50:  700nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50240865(CHEMBL157844 | (4aS,6aS,12aR,12bS)-10-Hydroxy-4,4,...)
Affinity DataEC50:  3.30E+3nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398328(CHEMBL2177348)
Affinity DataEC50:  2.70E+3nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398329(CHEMBL2177347)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398330(XESTOQUINONE)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50398331(MIMOSAMYCIN)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of HIF2alpha in human 786-0 cells expressing truncated HIF1alpha assessed as reduction in luciferase activity after 24 hrs by reporter gen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed