Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50040024
TargetLysophosphatidic acid receptor 5(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50388091(CHEMBL2058156)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human recombinant LPA5 receptor expressed in rat RH7777 cells assessed as inhibition of hexadecyl-LPA-induced effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 5(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50388091(CHEMBL2058156)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at LPA5 receptor in human washed platelets assessed as inhibition of hexadecyl-LPA-induced platelet aggregation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 5(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50388091(CHEMBL2058156)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at LPA5 receptor in human isolated platelets assessed as inhibition of hexadecyl-LPA-induced platelet aggregation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50388091(CHEMBL2058156)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at LPA2 receptor in human isolated platelets assessed as inhibition of TRAP-induced platelet aggregation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 5(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at LPA5 receptor in human isolated platelets assessed as inhibition of hexadecyl-LPA-induced platelet aggregation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 5(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50373826(CHEMBL256470)
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at LPA5 receptor in human isolated platelets assessed as inhibition of hexadecyl-LPA-induced platelet aggregation after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed