Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50039508
LigandPNGBDBM50305083(Ko143 | Ko-143 | 3-((3S,6S)-6-Isobutyl-9-methoxy-1...)
Affinity DataIC50: 50nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50379211(CHEMBL2011288)
Affinity DataIC50: 110nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50379213(CHEMBL2011290)
Affinity DataIC50: 160nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50379209(CHEMBL2011282)
Affinity DataIC50: 170nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50379208(CHEMBL2011287)
Affinity DataIC50: 180nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50379212(CHEMBL2011289)
Affinity DataIC50: 200nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50379210(CHEMBL2011286)
Affinity DataIC50: 470nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50305083(Ko143 | Ko-143 | 3-((3S,6S)-6-Isobutyl-9-methoxy-1...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MRP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed