Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50032889
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336217(4-chloro-N-(3-methoxyphenyl)-3-nitrobenzamide | CH...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336226(N-(3-methoxyphenyl)-3-nitro-4-(propylamino)benzami...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336224(4-(benzylamino)-N-(3-methoxyphenyl)-3-nitrobenzami...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336221(N-(3-methoxyphenyl)-3-nitro-4-(pyrrolidin-1-yl)ben...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336220(N-(3-methoxyphenyl)-3-nitro-4-(piperidin-1-yl)benz...)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336208(N-(3-fluorophenyl)-4-(pyrrolidin-1-yl)-3-(trifluor...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336210(N-(3-isopropoxyphenyl)-4-(pyrrolidin-1-yl)-3-(trif...)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336216(4-bromo-N-(3-methoxyphenyl)-3-nitrobenzamide | CHE...)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336228(N-(3-methoxyphenyl)-4-(4-methylpiperidin-1-yl)-3-n...)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336214(N-(3-methoxyphenyl)-4-(pyrrolidin-1-yl)-3-(trifluo...)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336215(4-(pyrrolidin-1-yl)-N-m-tolyl-3-(trifluoromethyl)b...)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336227(4-(ethylamino)-N-(3-methoxyphenyl)-3-nitrobenzamid...)
Affinity DataIC50: 75nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336219(N-(3-methoxyphenyl)-4-morpholino-3-nitrobenzamide ...)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336209(N-(3-acetylphenyl)-4-(pyrrolidin-1-yl)-3-(trifluor...)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336225(4-(isopropylamino)-N-(3-methoxyphenyl)-3-nitrobenz...)
Affinity DataIC50: 142nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336223(N-(3-methoxyphenyl)-3-nitro-4-(phenylamino)benzami...)
Affinity DataIC50: 175nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336213(N-(3-(difluoromethoxy)phenyl)-4-(pyrrolidin-1-yl)-...)
Affinity DataIC50: 187nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336222(4-(azetidin-1-yl)-N-(3-methoxyphenyl)-3-nitrobenza...)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336207(N-(3-chlorophenyl)-4-(pyrrolidin-1-yl)-3-(trifluor...)
Affinity DataIC50: 245nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336211(4-(pyrrolidin-1-yl)-N-(3-(1,1,2,2-tetrafluoroethox...)
Affinity DataIC50: 364nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336212(N-(3-ethylphenyl)-4-(pyrrolidin-1-yl)-3-(trifluoro...)
Affinity DataIC50: 470nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336206(N-(3-bromophenyl)-4-(pyrrolidin-1-yl)-3-(trifluoro...)
Affinity DataIC50: 568nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336218(N-(3-methoxyphenyl)-3-nitrobenzamide | CHEMBL16696...)
Affinity DataIC50: 665nMAssay Description:Antagonist activity at mouse TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336228(N-(3-methoxyphenyl)-4-(4-methylpiperidin-1-yl)-3-n...)
Affinity DataIC50: 3.79E+3nMAssay Description:Antagonist activity at human TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataIC50: 4.54E+3nMAssay Description:Antagonist activity at rat TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataIC50: 7.49E+3nMAssay Description:Antagonist activity at human TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human TAAR1 assessed as reversal of endogenous beta-PEA effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336205((N-(3-Ethoxy-phenyl)-4-pyrrolidin-1-yl-3-trifluoro...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336228(N-(3-methoxyphenyl)-4-(4-methylpiperidin-1-yl)-3-n...)
Affinity DataKi:  2nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336214(N-(3-methoxyphenyl)-4-(pyrrolidin-1-yl)-3-(trifluo...)
Affinity DataKi:  3nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336226(N-(3-methoxyphenyl)-3-nitro-4-(propylamino)benzami...)
Affinity DataKi:  4nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336229((+/-)-4-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-flu...)
Affinity DataKi:  4nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336210(N-(3-isopropoxyphenyl)-4-(pyrrolidin-1-yl)-3-(trif...)
Affinity DataKi:  4nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336224(4-(benzylamino)-N-(3-methoxyphenyl)-3-nitrobenzami...)
Affinity DataKi:  5nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336208(N-(3-fluorophenyl)-4-(pyrrolidin-1-yl)-3-(trifluor...)
Affinity DataKi:  9nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336213(N-(3-(difluoromethoxy)phenyl)-4-(pyrrolidin-1-yl)-...)
Affinity DataKi:  12nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336225(4-(isopropylamino)-N-(3-methoxyphenyl)-3-nitrobenz...)
Affinity DataKi:  12nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336220(N-(3-methoxyphenyl)-3-nitro-4-(piperidin-1-yl)benz...)
Affinity DataKi:  12nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336221(N-(3-methoxyphenyl)-3-nitro-4-(pyrrolidin-1-yl)ben...)
Affinity DataKi:  13nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336215(4-(pyrrolidin-1-yl)-N-m-tolyl-3-(trifluoromethyl)b...)
Affinity DataKi:  16nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336207(N-(3-chlorophenyl)-4-(pyrrolidin-1-yl)-3-(trifluor...)
Affinity DataKi:  20nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336212(N-(3-ethylphenyl)-4-(pyrrolidin-1-yl)-3-(trifluoro...)
Affinity DataKi:  21nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336216(4-bromo-N-(3-methoxyphenyl)-3-nitrobenzamide | CHE...)
Affinity DataKi:  21nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336227(4-(ethylamino)-N-(3-methoxyphenyl)-3-nitrobenzamid...)
Affinity DataKi:  24nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336243(3,4-dichloro-N-(3-methoxyphenyl)benzamide | CHEMBL...)
Affinity DataKi:  25nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336209(N-(3-acetylphenyl)-4-(pyrrolidin-1-yl)-3-(trifluor...)
Affinity DataKi:  26nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336223(N-(3-methoxyphenyl)-3-nitro-4-(phenylamino)benzami...)
Affinity DataKi:  29nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetTrace amine-associated receptor 1(Mouse)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50336222(4-(azetidin-1-yl)-N-(3-methoxyphenyl)-3-nitrobenza...)
Affinity DataKi:  29nMAssay Description:Inhibition of mouse TAAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
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