Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50031320
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311095(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-hexylure...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic beta3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311121(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-(2-(naph...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311117(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-(4-isopr...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311092((S)-4-(3-hexylureido)-N-(4-(2-(2-hydroxy-3-(4-hydr...)
Affinity DataIC50: 13nMAssay Description:Displacement of [35S]MK0677 from human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311116(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-(4-ethyl...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311119(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-(4-tert-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311120(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-(naphtha...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311118(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-(4-butyl...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311096(N-(4-(2-(ethylamino)-2-methylpropyl)phenyl)-4-(3-h...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311092((S)-4-(3-hexylureido)-N-(4-(2-(2-hydroxy-3-(4-hydr...)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human GHS-R1a expressed in HEK293 cells assessed as inhibition of ghrelin-stimulated intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311095(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-hexylure...)
Affinity DataIC50: 46nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311114(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-m-tolylu...)
Affinity DataIC50: 69nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311115(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-p-tolylu...)
Affinity DataIC50: 77nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311109(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-heptylur...)
Affinity DataIC50: 97nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311098(N-(4-(3-aminopropyl)phenyl)-4-(3-hexylureido)benze...)
Affinity DataIC50: 108nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311111(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-benzylur...)
Affinity DataIC50: 128nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311112(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-phenethy...)
Affinity DataIC50: 138nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311113(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-o-tolylu...)
Affinity DataIC50: 161nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311108(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-pentylur...)
Affinity DataIC50: 241nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311110(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-phenylur...)
Affinity DataIC50: 263nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311094(N-(4-(2-aminoethyl)phenyl)-4-(3-hexylureido)benzen...)
Affinity DataIC50: 272nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311099(N-(4-(3-amino-3-methylbutyl)phenyl)-4-(3-hexylurei...)
Affinity DataIC50: 310nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311102(N-(3-(3-aminopropyl)phenyl)-4-(3-hexylureido)benze...)
Affinity DataIC50: 429nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311100(N-(4-(3-amino-2,2-dimethylpropyl)phenyl)-4-(3-hexy...)
Affinity DataIC50: 444nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311107(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-butylure...)
Affinity DataIC50: 474nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311101(N-(3-(2-aminoethyl)phenyl)-4-(3-hexylureido)benzen...)
Affinity DataIC50: 625nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311103(4-(3-hexylureido)-N-(4-(2-methyl-2-(2,2,2-trifluor...)
Affinity DataIC50: 682nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311106(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-isopropy...)
Affinity DataIC50: 846nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311105(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-propylur...)
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311097(N-(4-(aminomethyl)phenyl)-4-(3-hexylureido)benzene...)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311093(4-(3-hexylureido)-N-phenylbenzenesulfonamide | CHE...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311095(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-hexylure...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human adrenergic beta3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50311104(N-(4-(2-amino-2-methylpropyl)phenyl)-4-(3-ethylure...)
Affinity DataIC50: 5.62E+3nMAssay Description:Inhibition of human GHS-R1aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed