Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50036865
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 0.900nMAssay Description:Tested for binding affinity against H197A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 1.10nMAssay Description:Tested for binding affinity against H265A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 1.40nMAssay Description:Tested for binding affinity against human wild type NK1 receptor expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 1.70nMAssay Description:Tested for binding affinity against Q165A mutant NK1 receptor expressed in CHO cells, using [125]SP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409025(CHEMBL2112246)
Affinity DataIC50: 27nMAssay Description:Tested for binding affinity against Tachykinin receptor 2 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369642(CHEMBL1790897)
Affinity DataIC50: 28nMAssay Description:Tested for binding affinity against Tachykinin receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369645(CHEMBL1790894)
Affinity DataIC50: 44nMAssay Description:Tested for binding affinity against Tachykinin receptor 1 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409026(CHEMBL2112245)
Affinity DataIC50: 46nMAssay Description:Tested for binding affinity against Tachykinin receptor 2 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369646(CHEMBL1790896)
Affinity DataIC50: 100nMAssay Description:Tested for binding affinity against human somatostatin receptor subtype 4 (hSSTR4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50051567(5-{(2R,3R,4S,5R,6R)-3,4,5-Tris-benzyloxy-6-[2-(1H-...)
Affinity DataIC50: 120nMAssay Description:Tested for binding affinity against Tachykinin receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409025(CHEMBL2112246)
Affinity DataIC50: 220nMAssay Description:Tested for binding affinity against Tachykinin receptor 1 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409025(CHEMBL2112246)
Affinity DataIC50: 240nMAssay Description:Tested for binding affinity against human wild type NK1 receptor expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409026(CHEMBL2112245)
Affinity DataIC50: 250nMAssay Description:Tested for binding affinity against Tachykinin receptor 1 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409026(CHEMBL2112245)
Affinity DataIC50: 260nMAssay Description:Tested for binding affinity against human wild type NK1 receptor expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369645(CHEMBL1790894)
Affinity DataIC50: 730nMAssay Description:Tested for binding affinity against Tachykinin receptor 2 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369644(CHEMBL1790895)
Affinity DataIC50: 850nMAssay Description:Tested for binding affinity against Tachykinin receptor 2 expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409026(CHEMBL2112245)
Affinity DataIC50: 900nMAssay Description:Tested for binding affinity against H197A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409025(CHEMBL2112246)
Affinity DataIC50: 950nMAssay Description:Tested for binding affinity against H197A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369645(CHEMBL1790894)
Affinity DataIC50: 1.40E+3nMAssay Description:Tested for binding affinity against human wild type NK1 receptor expressed in CHO cells, using [125]SP as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369645(CHEMBL1790894)
Affinity DataIC50: 2.70E+3nMAssay Description:Tested for binding affinity against H197A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369645(CHEMBL1790894)
Affinity DataIC50: 3.60E+3nMAssay Description:Tested for binding affinity against Q165A mutant NK1 receptor expressed in CHO cells, using [125]SP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409025(CHEMBL2112246)
Affinity DataIC50: 6.10E+3nMAssay Description:Tested for binding affinity against H265A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50369645(CHEMBL1790894)
Affinity DataIC50: 8.20E+3nMAssay Description:Tested for binding affinity against H265A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50409026(CHEMBL2112245)
Affinity DataIC50: 9.60E+3nMAssay Description:Tested for binding affinity against H265A mutant NK1 receptor using [125]SP radioligand in COS cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed