Compile Data Set for Download or QSAR
Report error Found 2053 of ic50 data for polymerid = 999
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50236330(CHEMBL4070196)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447747(CHEMBL3113272)
Affinity DataIC50: 0.170nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359728([3-(3-carbamoylphenyl)-5- fluoro-phenyl]N- cyclohe...)
Affinity DataIC50: 0.230nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359728([3-(3-carbamoylphenyl)-5- fluoro-phenyl]N- cyclohe...)
Affinity DataIC50: 0.230nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50295654(Dodecylcarbamic acid 3-(1,2,3-thiadiazol-4-yl)phen...)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of FAAH in Wistar rat cerebral membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447746(CHEMBL3113273)
Affinity DataIC50: 0.280nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50437233(CHEMBL2402911)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Wistar rat brain FAAH using [3H]-ethanolamine as substrate preincubated for 20 mins followed by substrate addition by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50236334(CHEMBL4071240)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50551026(CHEMBL4749527)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM23316(7-phenyl-1-{pyrido[2,3-d][1,3]oxazol-2-yl}heptan-1...)
Affinity DataIC50: 0.316nMpH: 9.0 T: 2°CAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [3H]anandamide was evaluated by using rat brain homogenate preparations. [3H]Ethanola...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50419129(CHEMBL1830441)
Affinity DataIC50: 0.331nMAssay Description:Displacement of [3H]-anandamide from rat brain FAAH after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447745(CHEMBL3113274)
Affinity DataIC50: 0.340nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50458983(CHEMBL4207166)
Affinity DataIC50: 0.360nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50434329(CHEMBL2386554)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447749(CHEMBL3113270)
Affinity DataIC50: 0.430nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50458984(CHEMBL4218897)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50426652(CHEMBL2326178)
Affinity DataIC50: 0.460nMAssay Description:Apparent inhibition of rat FAAH after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50437231(CHEMBL2402925)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Wistar rat brain FAAH using [3H]-ethanolamine as substrate preincubated for 20 mins followed by substrate addition by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50437232(CHEMBL2402921 | 3‐(3‐carbamoylphenyl)&...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Wistar rat brain FAAH using [3H]-ethanolamine as substrate preincubated for 20 mins followed by substrate addition by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of rat intact neuron FAAHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FAAH in Wistar rat brain intact neurons assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50424227(CHEMBL2314112)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 90 mins prior to ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50434318(CHEMBL2386566)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50271030(Naphthalen-2-ylmethylcarbamic Acid 3'-Carbamoylbip...)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of FAAH in rat brain membrane assessed as [3H]anandamide hydrolysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50458981(CHEMBL4206642)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50271030(Naphthalen-2-ylmethylcarbamic Acid 3'-Carbamoylbip...)
Affinity DataIC50: 0.631nMAssay Description:Displacement of [3H]-anandamide from rat brain FAAH after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM23078(CHEMBL227046 | 3-(4-phenylphenyl)-1-[5-(pyridin-2-...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of rat recombinant FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50402675(CHEMBL2207348)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of rat FAAH preincubated for 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359718([4-fluoro-3-(3- sulfamoylphenyl)phenyl] N-cyclohex...)
Affinity DataIC50: 0.700nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359718([4-fluoro-3-(3- sulfamoylphenyl)phenyl] N-cyclohex...)
Affinity DataIC50: 0.700nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50551011(CHEMBL4781803)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50426650(CHEMBL2326177)
Affinity DataIC50: 0.710nMAssay Description:Apparent inhibition of rat FAAH after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50426651(CHEMBL2326194)
Affinity DataIC50: 0.75nMAssay Description:Apparent inhibition of rat FAAH after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50426648(CHEMBL2326197)
Affinity DataIC50: 0.800nMAssay Description:Apparent inhibition of rat FAAH after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50551027(CHEMBL4752215)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50436356(CHEMBL2396702)
Affinity DataIC50: 0.813nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50436356(CHEMBL2396702)
Affinity DataIC50: 0.820nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate preincubated for 60 mins by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50458979(CHEMBL4210086)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359719([3-(3-carbamoylphenyl)-4- fluoro-phenyl]N- cyclobu...)
Affinity DataIC50: 0.900nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359719([3-(3-carbamoylphenyl)-4- fluoro-phenyl]N- cyclobu...)
Affinity DataIC50: 0.900nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50426649(CHEMBL2326192)
Affinity DataIC50: 0.960nMAssay Description:Apparent inhibition of rat FAAH after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50228837(2-(3-biphenyl-4-yl-propionyl)-oxazole-5-carbonitri...)
Affinity DataIC50: 1nMAssay Description:Inhibition of rat recombinant FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50161511(1-(5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl)-heptan-1-o...)
Affinity DataIC50: 1nMAssay Description:Inhibition of rat FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50262135(1-(1,3,4-Oxadiazol-2-yl)-7-phenylheptan-1-one | CH...)
Affinity DataIC50: 1nMAssay Description:Inhibition of rat FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50437230(CHEMBL2402922)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Wistar rat brain FAAH using [3H]-ethanolamine as substrate preincubated for 20 mins followed by substrate addition by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50298655(3-(4,5-Dihydrooxazol-2-yl)phenyl cyclohexylcarbama...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FAAH in Wistar rat brain assessed as by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447748(CHEMBL3113271)
Affinity DataIC50: 1.20nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50424227(CHEMBL2314112)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of FAAH-mediated [3H]anandamide hydrolysis in rat brain homogenate assessed as [3H]ethanolamine production incubated for 45 mins prior to ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50426645(CHEMBL2326193)
Affinity DataIC50: 1.20nMAssay Description:Apparent inhibition of rat FAAH after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50434314(CHEMBL2386570)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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