Compile Data Set for Download or QSAR
Report error Found 35 of ic50 data for polymerid = 9750
LigandPNGBDBM50526770(CHEMBL4519504)
Affinity DataIC50: 5nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50236530(CHEMBL3727577)
Affinity DataIC50: 26nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236530(CHEMBL3727577)
Affinity DataIC50: 40nMAssay Description:Inhibition of PDHK3 (unknown origin) assessed as decrease in phosphorylation of E1alpha subunit at serine 293 residue after 1 hr by DELFIAMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50526757(CHEMBL4575355)
Affinity DataIC50: 59nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526772(CHEMBL4461160)
Affinity DataIC50: 64nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526758(CHEMBL4570690)
Affinity DataIC50: 67nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526756(CHEMBL4591977)
Affinity DataIC50: 80nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526780(CHEMBL4551410)
Affinity DataIC50: 90nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526759(CHEMBL4452536)
Affinity DataIC50: 90nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526771(CHEMBL4513465)
Affinity DataIC50: 98nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50236530(CHEMBL3727577)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236530(CHEMBL3727577)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50526774(CHEMBL4540811)
Affinity DataIC50: 136nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526777(CHEMBL4434941)
Affinity DataIC50: 142nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526769(CHEMBL4587341)
Affinity DataIC50: 181nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526773(CHEMBL4558944)
Affinity DataIC50: 186nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526784(CHEMBL4558837)
Affinity DataIC50: 255nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526764(CHEMBL4561336)
Affinity DataIC50: 461nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50526768(CHEMBL4579724)
Affinity DataIC50: 858nMAssay Description:Inhibition of PDHK3 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50232913(CHEMBL4103350)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of recombinant human PDK3 in presence of E1 protein and PDC core E2/E3BP incubated for 10 mins by titration assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM227593(PS8)
Affinity DataIC50: 2.55E+3nMpH: 7.5 T: 2°CAssay Description:To determine the IC50 for PDK inhibitors, a mixture containing 0.05-0.2 μM PDK, 6μM E1, with or without 0.5 μM of the PDC core E2/E3BP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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LigandPNGBDBM50529881(CHEMBL4434895)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
LigandPNGBDBM50529881(CHEMBL4434895)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50032655(CHEMBL3354665)
Affinity DataIC50: 5.34E+3nMAssay Description:Inhibition of recombinant PDHK3 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50529878(CHEMBL4476534)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50529878(CHEMBL4476534)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50529879(CHEMBL4434775)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50529879(CHEMBL4434775)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of recombinant human His-tagged PDK3 expressed in Escherichia coli using PDH E1 as substrate measured after 30 mins by Kinase-Glo luminesc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50571960(CHEMBL4848983)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of human PDHK3 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrate preincubated with enzyme complex for 45...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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LigandPNGBDBM227593(PS8)
Affinity DataIC50: 1.37E+4nMpH: 7.5 T: 2°CAssay Description:To determine the IC50 for PDK inhibitors, a mixture containing 0.05-0.2 μM PDK, 6μM E1, with or without 0.5 μM of the PDC core E2/E3BP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
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PubMed
LigandPNGBDBM227594(PS10)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of PDHK3 (unknown origin) assessed as decrease in phosphorylation of E1alpha subunit at serine 293 residue after 1 hr by DELFIAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM227594(PS10)
Affinity DataIC50: 2.13E+4nMpH: 7.5 T: 2°CAssay Description:To determine the IC50 for PDK inhibitors, a mixture containing 0.05-0.2 μM PDK, 6μM E1, with or without 0.5 μM of the PDC core E2/E3BP...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50232913(CHEMBL4103350)
Affinity DataIC50: 4.58E+4nMAssay Description:Inhibition of recombinant human PDK3 in presence of E1 protein incubated for 10 mins by titration assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50347503(RADICICOL)
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibition of PDHK3 (unknown origin)More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM227588(DCA)
Affinity DataIC50: 5.56E+6nMAssay Description:Inhibition of PDK3 (unknown origin) using full length His6-tagged PDHA1 as substrate after 30 mins by ELISAMore data for this Ligand-Target Pair
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PubMed