Compile Data Set for Download or QSAR
Report error Found 48 of ic50 data for polymerid = 9125,49000212,49000216,49000218,49000229,49000231,49000232
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403738(CHEMBL351483)
Affinity DataIC50: 0.955nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403739(CHEMBL163247)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403740(CHEMBL165350)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403755(CHEMBL163190)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403752(CHEMBL162370)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403747(CHEMBL162826)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403746(CHEMBL162147)
Affinity DataIC50: 1.90nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403745(CHEMBL162490)
Affinity DataIC50: 2nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403753(CHEMBL162682)
Affinity DataIC50: 2.10nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403750(CHEMBL351200)
Affinity DataIC50: 2.10nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403748(CHEMBL162232)
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403742(CHEMBL165796)
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403744(LUSAPERIDONE)
Affinity DataIC50: 2.60nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403751(CHEMBL162436)
Affinity DataIC50: 4.20nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403754(CHEMBL164612)
Affinity DataIC50: 4.40nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403749(CHEMBL165181)
Affinity DataIC50: 11nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403737(CHEMBL165776)
Affinity DataIC50: 11nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
Bayer

Curated by ChEMBL
LigandPNGBDBM50632390(CHEMBL5410211)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at rat adrenergic alpha2BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataIC50: 19nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Dog)
Bayer

Curated by ChEMBL
LigandPNGBDBM50632390(CHEMBL5410211)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at dog adrenergic alpha2BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403741(CHEMBL165677)
Affinity DataIC50: 79nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50403743(CHEMBL162058)
Affinity DataIC50: 195nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50115644((+/-)-12-Methyl-1,2,3,4,9,13b-hexahydro-2,4a,5-tri...)
Affinity DataIC50: 224nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626148(US11786528, Example 35)
Affinity DataIC50: 530nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626022(US11786528, Example 11)
Affinity DataIC50: 580nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Rat)
Bayer

Curated by ChEMBL
LigandPNGBDBM50083342(7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-4H-be...)
Affinity DataIC50: 630nMAssay Description:Inhibition of [3H]- Yohimbine binding against rat kidney cortex Alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626015(US11786528, Example 10)
Affinity DataIC50: 690nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50244809((2R)-2-[3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(triflu...)
Affinity DataIC50: 770nMAssay Description:Displacement of radioligand from adrenergic alpha2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50511341(CHEMBL4483761)
Affinity DataIC50: 790nMAssay Description:Displacement of [3H]RX 821002 from human recombinant adrenergic alpha-2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50065660(CHEMBL3403995)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of alpha-adrenoceptor 2B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50174702((R)-N-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human adrenergic alpha-2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626057(US11786528, Example 19)
Affinity DataIC50: 1.45E+3nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626180(US11786528, Example 40)
Affinity DataIC50: 1.46E+3nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM625944(2-[(3-methylphenyl)methyl]-6-(1,2-thiazol-3-yl)-2H...)
Affinity DataIC50: 1.50E+3nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50026868(2-(1H-indol-3-yl)-N,N-dimethylethanamine | DMT | N...)
Affinity DataIC50: 1.58E+3nMAssay Description:Displacement of [3H]-rauwolscine from human recombinant adrenergic alpha-2b receptor expressed in human CHO-K1 cells incubated for 60 mins by spectro...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50026868(2-(1H-indol-3-yl)-N,N-dimethylethanamine | DMT | N...)
Affinity DataIC50: 1.67E+3nMAssay Description:Displacement of [3H]-rauwolscine from human recombinant adrenergic alpha-2b receptor expressed in human CHO-K1 cells incubated for 60 mins by spectro...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50092139(CHEMBL3582472)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of adrenergic alpha-2B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM625941(US11786528, Comparative Example 1)
Affinity DataIC50: 4.91E+3nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50319673(1-[6-(4-Fluorophenyl)pyridin-3-yl]-3-(4-piperidin-...)
Affinity DataIC50: 7.50E+3nMAssay Description:Binding affinity to adrenergic alpha2B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50240277(CHEMBL4061793)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at human alpha2B-adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626028(US11786528, Example 12)
Affinity DataIC50: 9.00E+3nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50212239(5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H](-)CGP-12177 from adrenergic beta2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50318666(NITD609 | (1R,3S)-5',7-Dichloro-6-fluoro-3-methyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human recombinant alpha2b receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50304075(3-(5-(4-tert-butylphenyl)-3-((dimethylamino)methyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alpha2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626170(US11786528, Example 38)
Affinity DataIC50: 1.17E+4nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626100(US11786528, Example 24)
Affinity DataIC50: 2.56E+4nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM50401271(CHEMBL2203713 | CHEMBL3216328)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of alpha2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Janssen Research Foundation

Curated by ChEMBL
LigandPNGBDBM626206(US11786528, Example 46)
Affinity DataIC50: 1.00E+5nMAssay Description:Affinity for the human adenosine receptor sub-types (A2a, A2b, A1 and A3) was determined by SPR as described in Aristotelous, T., et al, Methods in E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent