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Report error Found 3 of ic50 data for polymerid = 8933
TargetSerine/threonine-protein kinase PAK 1 [249-545,K299R](Human)
The Scripps Research Institute

LigandPNGBDBM50112347(CHEMBL3609327 | FRAX597)
Affinity DataIC50: 7.70nMAssay Description:IC50 values were determined using a 10 concentration point, non-radioactive, functional assay that employs a fluorescence-based, coupled enzyme forma...More data for this Ligand-Target Pair
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PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 1 [249-545,K299R](Human)
The Scripps Research Institute

LigandPNGBDBM213235(FRAX414)
Affinity DataIC50: 20nMAssay Description:IC50 values were determined using a 10 concentration point, non-radioactive, functional assay that employs a fluorescence-based, coupled enzyme forma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetSerine/threonine-protein kinase PAK 1 [249-545,K299R](Human)
The Scripps Research Institute

LigandPNGBDBM6276(Pyrido[2,3-d]pyrimidin-7-one 1 | 8-Cyclopentyl-2-[...)
Affinity DataIC50: 483nMAssay Description:IC50 values were determined using a 10 concentration point, non-radioactive, functional assay that employs a fluorescence-based, coupled enzyme forma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed