Compile Data Set for Download or QSAR
Report error Found 11 of ic50 data for polymerid = 802
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50246253(AZD-5438 | 4-(1-isopropyl-2-methyl-1H-imidazol-5-y...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Cyclin E/CDK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59097(Aminopyrimidine, 10)
Affinity DataIC50: 220nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)
Affinity DataIC50: 230nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59092(Aminopyrimidine, 2)
Affinity DataIC50: 330nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59091(Aminopyrimidine, 1)
Affinity DataIC50: 410nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59093(Aminopyrimidine, 3)
Affinity DataIC50: 430nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59095(Aminopyrimidine, 7)
Affinity DataIC50: 1.02E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59094(Aminopyrimidine, 6)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50319619(Aminopyrimidine, 5 | CHEMBL1085626 | 4-(2,4-Dimeth...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG1/S-specific cyclin-E1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM59096(Aminopyrimidine, 8)
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro kinase inhibition assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed