Compile Data Set for Download or QSAR
Report error Found 874 of ic50 data for polymerid = 7859,50006569
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50169057(CHEMBL3805896)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50169056(CHEMBL3806163)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435435(US10570116, Compound C43)
Affinity DataIC50: 0.230nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50169061(CHEMBL3805393)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50544641(CHEMBL4645574)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50544643(CHEMBL4634919)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435441(US10570116, Compound C49)
Affinity DataIC50: 0.300nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435395(US10570116, Compound C6)
Affinity DataIC50: 0.310nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435386(US10570116, Compound C2)
Affinity DataIC50: 0.320nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435444(US10570116, Compound C52)
Affinity DataIC50: 0.330nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435439(US10570116, Compound C47)
Affinity DataIC50: 0.350nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50544640(CHEMBL4640008)
Affinity DataIC50: 0.360nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50169060(CHEMBL3804939)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50544645(CHEMBL4643690)
Affinity DataIC50: 0.410nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435431(US10570116, Compound C39)
Affinity DataIC50: 0.430nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435442(US10570116, Compound C50)
Affinity DataIC50: 0.440nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435434(US10570116, Compound C42)
Affinity DataIC50: 0.450nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435437(US10570116, Compound C45)
Affinity DataIC50: 0.450nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435409(US10570116, Compound C17)
Affinity DataIC50: 0.470nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435426(US10570116, Compound C34)
Affinity DataIC50: 0.480nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435399(US10570116, Compound C8)
Affinity DataIC50: 0.5nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50544644(CHEMBL4639702)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435425(US10570116, Compound C33)
Affinity DataIC50: 0.510nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435403(US10570116, Compound C11)
Affinity DataIC50: 0.520nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50544642(CHEMBL4632401)
Affinity DataIC50: 0.520nMAssay Description:Inhibition of human GST-tagged tankyrase 1 autophosphorylation by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435384(US10570116, Compound C1)
Affinity DataIC50: 0.570nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435410(US10570116, Compound C18)
Affinity DataIC50: 0.580nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435430(US10570116, Compound C38)
Affinity DataIC50: 0.580nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435433(US10570116, Compound C41)
Affinity DataIC50: 0.590nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50593627(CHEMBL5199558)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 - 1327 residues) (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50593627(CHEMBL5199558)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate assessed as inhibition of autoPARsylation activity incubated for 1 hr by ELI...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435408(US10570116, Compound C16)
Affinity DataIC50: 0.610nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435422(US10570116, Compound C30)
Affinity DataIC50: 0.620nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435396(US10570116, Compound C7)
Affinity DataIC50: 0.660nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435424(US10570116, Compound C32)
Affinity DataIC50: 0.680nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435428(US10570116, Compound C36)
Affinity DataIC50: 0.790nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50505331(CHEMBL4458129)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of GST tagged-TEV cleavage site-fused human recombinant TNKS1 (1023 to 1327 residues) expressed in baculovirus infected sf9 cells assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50620061(CHEMBL5401025)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50409622(CHEMBL5272750)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate assessed as inhibition of autoPARsylation activity incubated for 1 hr by ELI...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50409634(CHEMBL5274873)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate assessed as inhibition of autoPARsylation activity incubated for 1 hr by ELI...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50169058(CHEMBL3806049)
Affinity DataIC50: 0.810nMAssay Description:Inhibition of GST-tagged TNKS1 (1023 to 1327 residues) (unknown origin) autoparsylation using biotinylated NAD incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435393(US10570116, Compound C4)
Affinity DataIC50: 0.840nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435412(US10570116, Compound C20)
Affinity DataIC50: 0.920nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435429(US10570116, Compound C37)
Affinity DataIC50: 0.950nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435443(US10570116, Compound C51)
Affinity DataIC50: 1nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50188594(CHEMBL1086580 | CHEBI:62878 | US20240279201, Compo...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged TNKS1 (1001 to 1327(end) residues) expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50409619(CHEMBL5271127)
Affinity DataIC50: 1nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate assessed as inhibition of autoPARsylation activity incubated for 1 hr by ELI...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50094926(CHEMBL3589282)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human TNKS1 catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM435445(US10570116, Compound C53)
Affinity DataIC50: 1.10nMAssay Description:TNKS 1 and 2: The activity ELISA is performed in 384 well Glutathione coated microtiter plates (Express capture Glutathione coated plate, Biocat, Hei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50505324(CHEMBL4588170)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of GST tagged-TEV cleavage site-fused human recombinant TNKS1 (1023 to 1327 residues) expressed in baculovirus infected sf9 cells assessed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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