Compile Data Set for Download or QSAR
Report error Found 13 of ic50 data for polymerid = 7813
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50: 17nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM50420459(CHEMBL2086528)
Affinity DataIC50: 840nMAssay Description:Inhibition of human recombinant TG6 by fluorescent transamidation assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: 2.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: 5.00E+3nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50392881(CHEMBL2152090)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human TGM6More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM185182([2-[[2-[4-[[5-(Dimethylamino)-1-naphthyl]sulfonyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM185172([2-[[2-[4-(Adamantane-1-carbonyl)piperazin-1-yl]-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM185177(1-Adamantylmethyl 4-[2-(prop-2-enoylamino)acetyl]p...)
Affinity DataIC50: 1.00E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50392906(CHEMBL2152204)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of human TGM6More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50400625(CHEMBL2203469)
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of transglutaminase 6More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50400619(CHEMBL2203476)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of transglutaminase 6More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50400621(CHEMBL2203451)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of transglutaminase 6More data for this Ligand-Target Pair
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PubMed