Compile Data Set for Download or QSAR
Report error Found 844 of ic50 data for polymerid = 7501,50003883,50007938
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50485288(CHEMBL2046980)
Affinity DataIC50: 0.00150nMAssay Description:Inhibition of HIV1 3B protease activity in human H9 cells using Abz-Thr-Ile-Nle-Phe(p-NO2)-Gln-Arg-NH2 as substrate after 40 mins by spectrophotometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482331(CHEMBL1170704)
Affinity DataIC50: 0.00700nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50280116(CHEMBL4177355)
Affinity DataIC50: 0.0120nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using Val-Ser-Gln-Asn-(beta-naphtyl)Ala-Pro-Ile-Val as substrate preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM8125(Darunavir (DRV) | CHEMBL1323 | (3R,3aS,6aR)-hexahy...)
Affinity DataIC50: 0.0130nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using Val-Ser-Gln-Asn-(beta-naphtyl)Ala-Pro-Ile-Val as substrate preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482336(CHEMBL1170709)
Affinity DataIC50: 0.0130nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482332(CHEMBL1170706)
Affinity DataIC50: 0.0160nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482337(CHEMBL1170703)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50127975((R)-N-(2,6-dimethylbenzyl)-3-((2S,4R)-4-benzyl-2-h...)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM13934(CGP 73547 | CHEMBL1163 | methyl N-[(1S)-1-{[(2S,3S...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of wild-type HIV1 protease expressed in Escherichia coli assessed as reduction in product formation preincubated for 30 mins followed by a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM13934(CGP 73547 | CHEMBL1163 | methyl N-[(1S)-1-{[(2S,3S...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using Val-Ser-Gln-Asn-(beta-naphtyl)Ala-Pro-Ile-Val as substrate preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50497089(CHEMBL3263091)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of purified HIV-1 protease using [Arg-Glu(EDANS)-Ser-Gin-Asn-Tyr-Ile-Val-Gin-Lys(dabcyl)-Arg) as fluorogenic substrate by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM8125(Darunavir (DRV) | CHEMBL1323 | (3R,3aS,6aR)-hexahy...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using Arg-Glu (EDANS)-Ser-GlnAsn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincuba...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM8125(Darunavir (DRV) | CHEMBL1323 | (3R,3aS,6aR)-hexahy...)
Affinity DataIC50: 0.0610nMT: 2°CAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli incubated for 20 to 30 mins at room temperature using (Arg-Glu(EDANS)-Ser-Gln-Asn-Tyr-Pro-I...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478722(KNI-1933 | CHEMBL452953)
Affinity DataIC50: 0.0830nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478719(KNI-1965 | CHEMBL509400)
Affinity DataIC50: 0.0860nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478712(KNI-1969 | CHEMBL485911)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478713(KNI-1961 | CHEMBL510136)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50497086(CHEMBL3263090)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of purified HIV-1 protease using [Arg-Glu(EDANS)-Ser-Gin-Asn-Tyr-Ile-Val-Gin-Lys(dabcyl)-Arg) as fluorogenic substrate by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482333(CHEMBL1170707)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482334(CHEMBL1170708)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50477633(CHEMBL398053)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50477640(CHEMBL247616)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50497088(CHEMBL3263089)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of purified HIV-1 protease using [Arg-Glu(EDANS)-Ser-Gin-Asn-Tyr-Ile-Val-Gin-Lys(dabcyl)-Arg) as fluorogenic substrate by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50477636(CHEMBL395214)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478715(KNI-1910 | CHEMBL452873)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50497090(CHEMBL3263092)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of purified HIV-1 protease using [Arg-Glu(EDANS)-Ser-Gin-Asn-Tyr-Ile-Val-Gin-Lys(dabcyl)-Arg) as fluorogenic substrate by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50477638(CHEMBL397403)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50485183(CHEMBL2034991)
Affinity DataIC50: 0.170nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50477635(CHEMBL247615)
Affinity DataIC50: 0.170nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478721(KNI-1931 | CHEMBL230484)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50477634(CHEMBL395207)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of wild type HIV1 NL4-3 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478714(KNI-1909 | CHEMBL462726)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478718(KNI-1932 | CHEMBL455816)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478720(KNI-1960 | CHEMBL508278)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM13934(CGP 73547 | CHEMBL1163 | methyl N-[(1S)-1-{[(2S,3S...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481018(CHEMBL568883)
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481028(CHEMBL566620)
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481029(CHEMBL569671)
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481036(CHEMBL568589)
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481014(CHEMBL568951)
Affinity DataIC50: 0.339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50270566(CHEMBL4129828)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using Arg-Glu (EDANS)-Ser-GlnAsn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50497087(CHEMBL3263094)
Affinity DataIC50: 0.360nMAssay Description:Inhibition of purified HIV-1 protease using [Arg-Glu(EDANS)-Ser-Gin-Asn-Tyr-Ile-Val-Gin-Lys(dabcyl)-Arg) as fluorogenic substrate by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50478716(KNI-1878 | CHEMBL449836)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481020(CHEMBL565964)
Affinity DataIC50: 0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50481023(CHEMBL566849)
Affinity DataIC50: 0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50482338(CHEMBL1170705)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50067593(CHEBI:44032 | Crixivan | Indinavir | L-735524 | MK...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50213021(CHEBI:63621 | Fortovase | Invirase | Ro-31-8959 | ...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant wild type HIV1 protease assessed as hydrolysis of fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50497085(CHEMBL3263093)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of purified HIV-1 protease using [Arg-Glu(EDANS)-Ser-Gin-Asn-Tyr-Ile-Val-Gin-Lys(dabcyl)-Arg) as fluorogenic substrate by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtease(Human immunodeficiency virus type 1)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM8125(Darunavir (DRV) | CHEMBL1323 | (3R,3aS,6aR)-hexahy...)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli using Arg-Glu (EDANS)-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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