Report error Found 15 of ic50 data for polymerid = 7004
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 68nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 130nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 150nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 170nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 250 nM APAH (∼50% Zn2+ occupancy), 150 μM substrate, and 0−250 μM inhibit...More data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 270nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 390nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of Mycoplana ramosa acetylpolyamine amidohydrolase assessed as substrate deacetylation using L-Lys(epsilon-acetyl)-coumarin as substrate p...More data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 3.80E+5nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 1.90E+6nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
TargetAcetylpolyamine amidohydrolase(Mycoplana ramosa (Gram-negative bacterium))
University of Pennsylvania
University of Pennsylvania
Affinity DataIC50: 1.80E+6nMAssay Description:Inhibition of Mycoplana ramosa APAH expressed in Escherichia coli BL21 (DE3) using BML-KI104 as substrate after 30 mins by fluorimetric assayMore data for this Ligand-Target Pair
