Compile Data Set for Download or QSAR
Report error Found 234 of ic50 data for polymerid = 5442
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446884(CHEMBL3115282)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446883(CHEMBL3115283)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446882(CHEMBL3115284)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385803(CHEMBL2041190)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446887(CHEMBL3115295)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446903(CHEMBL3115293)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446902(CHEMBL3115294)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446901(CHEMBL3115296)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446904(CHEMBL3115292)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446905(CHEMBL3115291)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446906(CHEMBL3115290)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446907(CHEMBL3115289)
Affinity DataIC50: 1nMAssay Description:Inhibition of 6His-tagged PHD3 (1 to 239) (unknown origin)-mediated Cy5CODD hydroxylation expressed in Escherichia coli preincubated for 3 mins follo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50317545(CHEMBL4173371)
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD3 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50446903(CHEMBL3115293)
Affinity DataIC50: 1nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD3 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385806(CHEMBL2041193)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PHD3 (unknown origin) expressed in Sf9 cells using HIF-1alpha peptide as substrate preincubated for 30 mins followed by substrate addit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385788(CHEMBL2041175)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385806(CHEMBL2041193)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385806(CHEMBL2041193)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of FLAG- tagged full length HIF-PHD3 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385814(CHEMBL2043169)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385819(CHEMBL2043325)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385826(CHEMBL2041010)
Affinity DataIC50: 2nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385830(CHEMBL2041185)
Affinity DataIC50: 2nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385805(CHEMBL2041192)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385813(CHEMBL2043168)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385801(CHEMBL2041188)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385796(CHEMBL2041182)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385782(CHEMBL2041169)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385811(CHEMBL2043010)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385818(CHEMBL2043324)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385797(CHEMBL2041183)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM93422(PHD Inhibitor, 12{1,1,2})
Affinity DataIC50: 4.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385802(CHEMBL2041189)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385799(CHEMBL2041186)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507415(CHEMBL4451025)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM93419(PHD Inhibitor, 12{2,4,1})
Affinity DataIC50: 5.30nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50317547(CHEMBL4163812)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of PHD3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385820(CHEMBL2043326)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507408(CHEMBL4561977)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385825(CHEMBL2040897)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507409(CHEMBL4476576)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM93430(PHD Inhibitor, 12{2,1,2})
Affinity DataIC50: 6.40nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385778(CHEMBL2041164)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507419(CHEMBL4462855)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507407(CHEMBL4590677)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507421(CHEMBL4462741)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507406(CHEMBL4452218)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507411(CHEMBL4474474)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385812(CHEMBL2043011)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50385798(CHEMBL2041184)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of PHD3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50507424(CHEMBL4452138)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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