Compile Data Set for Download or QSAR
Report error Found 21 of ic50 data for polymerid = 5399
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human LOK using RLGRDKYKTLRQIRQ as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
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PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human LOK using RLGRDKYKTLRQIRQ as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM93207(Kinase inhibitor, 5)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM8226(3-[(3-chlorophenyl)amino]-4-(2-methoxyphenyl)-2,5-...)
Affinity DataIC50: 12nMAssay Description:Inhibition of STK10 (unknown origin) expressed in Sf9 cells assessed as transfer of radiolabelled phosphate group from ATP by reaction biology methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM93207(Kinase inhibitor, 5)
Affinity DataIC50: 20nMpH: 7.5 T: 2°CAssay Description:Fluorescence assay used for determination of catch and release efficiency. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577328(CHEMBL4875188)
Affinity DataIC50: 23nMAssay Description:Inhibition of STK10 (unknown origin) expressed in Sf9 cells assessed as transfer of radiolabelled phosphate group from ATP by reaction biology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 52nMAssay Description:Inhibition of STK10More data for this Ligand-Target Pair
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PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577368(CHEMBL4878325)
Affinity DataIC50: 60nMAssay Description:Inhibition of STK10 (unknown origin) expressed in Sf9 cells assessed as transfer of radiolabelled phosphate group from ATP by reaction biology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577369(CHEMBL4856751)
Affinity DataIC50: 99nMAssay Description:Inhibition of STK10 (unknown origin) expressed in Sf9 cells assessed as transfer of radiolabelled phosphate group from ATP by reaction biology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM3175(Bisindolylmaleimide 11b | Ro 31-8220 | CHEMBL6291 ...)
Affinity DataIC50: 99nMAssay Description:Inhibition of STK10 (unknown origin) expressed in Sf9 cells assessed as transfer of radiolabelled phosphate group from ATP by reaction biology methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human STK10More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM8226(3-[(3-chlorophenyl)amino]-4-(2-methoxyphenyl)-2,5-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of biotinylated full-length STK10 expressed in Escherichia coli DH10Bac assessed as transfer of radiolabelled phosphate from ATP by OMNIA ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577340(CHEMBL4877889)
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of STK10 (unknown origin) expressed in Sf9 cells assessed as transfer of radiolabelled phosphate group from ATP by reaction biology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577328(CHEMBL4875188)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of biotinylated full-length STK10 expressed in Escherichia coli DH10Bac assessed as transfer of radiolabelled phosphate from ATP by OMNIA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577368(CHEMBL4878325)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of biotinylated full-length STK10 expressed in Escherichia coli DH10Bac assessed as transfer of radiolabelled phosphate from ATP by OMNIA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577369(CHEMBL4856751)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of biotinylated full-length STK10 expressed in Escherichia coli DH10Bac assessed as transfer of radiolabelled phosphate from ATP by OMNIA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50263167(3,4,5,6-Tetrahydro-2H-[1,2']bipyridinyl-4'-carboxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LOKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human LOK (1 to 348 residues) using RLGRDKYKTLRQI as substrate after 40 mins in presence of [gamma-33ATP] by radiometric sc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human LOK using [RLGRDKYKTLRQIRQ] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50429867(CHEMBL2333365)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LOK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50577340(CHEMBL4877889)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of biotinylated full-length STK10 expressed in Escherichia coli DH10Bac assessed as transfer of radiolabelled phosphate from ATP by OMNIA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed