Compile Data Set for Download or QSAR
Report error Found 51 of ic50 data for polymerid = 5007,50000097
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595287(CHEMBL5193958)
Affinity DataIC50: 130nMAssay Description:Inhibition of DPP3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595285(CHEMBL5175079)
Affinity DataIC50: 1.44E+3nMAssay Description:Competitive inhibition of DPP3 (unknown origin) using Arg-Arg-2-naphthylamide as substrateMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85267(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 1.70E+3nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85264(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 2.80E+3nM Kd:  200nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595281(CHEMBL5182137)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human DPP3 using Arg-Arg-2-naphthylamide as substrate assessed as reduction in release of 2-naphthylamine preincubated for 10 mins foll...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85265(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 5.60E+3nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85269(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 6.00E+3nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85268(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 7.00E+3nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595283(CHEMBL5187966)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of human DPP3 using Arg-Arg-2-naphthylamide as substrate assessed as reduction in release of 2-naphthylamine preincubated for 10 mins foll...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85270(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 8.00E+3nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595288(CHEMBL5199877)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of DPP3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85262(Benzimidazole derivative, 3)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85266(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85271(2,4-Disubstituted-1,3-di-(5-amidino-2-benzoimidazo...)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85261(Benzimidazole derivative, 2)
Affinity DataIC50: 1.80E+4nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595284(CHEMBL5176913)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human DPP3 using Arg-Arg-2-naphthylamide as substrate assessed as reduction in release of 2-naphthylamine preincubated for 10 mins foll...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 2.20E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595282(CHEMBL5191808)
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of human DPP3 using Arg-Arg-2-naphthylamide as substrate assessed as reduction in release of 2-naphthylamine preincubated for 10 mins foll...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50049391(norizalpinin | 3,5,7-trihydroxy-2-phenyl-4H-benzop...)
Affinity DataIC50: 2.34E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM7457(2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-chromen-4-on...)
Affinity DataIC50: 2.49E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50221073((3R,4S)-1-[6-(6-METHOXYPYRIDIN-3-YL)PYRIMIDIN-4-YL...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50249479(PF-00734200 | cis-(3,3-Difluoro-pyrrolidin-1-yl)-[...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3 in human erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187283((2R,5S)-1-(2-(1-(ethoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187258((2S,5R)-1-[2-(hexahydro-2,5-methano-pentalen-3a-yl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187266((2R,5S)-1-(2-(1-(hydroxymethyl)cyclopentylamino)ac...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187263((2S,5R)-1-[2-(3-hydroxy-adamantan-1-ylamino)-acety...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187275((2R,5S)-1-(2-(1-(methoxymethyl)cyclopentylamino)ac...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187268((2S,5R)-1-[2-(adamantan-1-ylamino)-acetyl]-pyrroli...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187261((2R,5S)-1-(2-(1-(butoxymethyl)cyclopentylamino)ace...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of DPP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM7462(cid_5280863 | CHEMBL150 | 3,5,7-trihydroxy-2-(4-hy...)
Affinity DataIC50: 3.29E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 3.66E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85260(Benzimidazole derivative, 1)
Affinity DataIC50: 5.30E+4nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM7458(Naringenin, 18 | 5,7-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataIC50: 5.40E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187657(3,6-dihydroxy-flavone | 3,6-dihydroxy-2-phenyl-4H-...)
Affinity DataIC50: 5.64E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50595286(CHEMBL5193133)
Affinity DataIC50: 7.40E+4nMAssay Description:Competitive inhibition of DPP3 (unknown origin) using Arg-Arg-2-naphthylamide as substrateMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 7.41E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50081950(6-hydroxy-2-phenyl-4H-chromen-4-one | NSC-26744 | ...)
Affinity DataIC50: 8.22E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM26658(2-(2,4-dihydroxyphenyl)-3,5,7-trihydroxychromen-4-...)
Affinity DataIC50: 8.50E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM26660(3,7-dihydroxy-2-phenyl-4H-chromen-4-one | CHEMBL21...)
Affinity DataIC50: 9.80E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM85263(Benzimidazole derivative, 4)
Affinity DataIC50: 1.00E+5nMpH: 7.4 T: 2°CAssay Description:The IC50 value is defined as the concentration of an inhibitor with caused 50% reduction of the enzyme activity under specific condition. The princi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM7461(5,7-dihydroxy-2-phenyl-4H-chromen-4-one | cid_5281...)
Affinity DataIC50: 1.23E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50187668(3-hydroxy-2-phenyl-4H-chromen-4-one | 3-Hydroxyfla...)
Affinity DataIC50: 1.88E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50174201(ARTHROTEC | GP 45840 | SOLARAZE | Sodium; [2-(2,6-...)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

TargetDipeptidyl peptidase 3(Human)
Graz University of Technology

Curated by ChEMBL
LigandPNGBDBM50028962(flavone | CHEMBL275638)
Affinity DataIC50: 2.93E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of flavonoids toward human DPP III was assayed in a 50 mM Tris-HCl buffer, pH 7.4. In brief, recombinant human DPP III (0.29 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM26197(Paracetamol | acetaminophen | CHEMBL112 | N-(4-hyd...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25756(Betalok | Spesikor | {2-hydroxy-3-[4-(2-methoxyeth...)
Affinity DataIC50: 3.15E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25758(2-hydroxy-5-{1-hydroxy-2-[(4-phenylbutan-2-yl)amin...)
Affinity DataIC50: 3.60E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM25753(Artrenolol | 2-{4-[2-hydroxy-3-(propan-2-ylamino)p...)
Affinity DataIC50: 3.75E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50056999(CHEMBL56367 | nimesulide)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

TargetDipeptidyl peptidase 3(wild yak)
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM22369(CHEMBL122 | MK 0966 | 4-(4-methanesulfonylphenyl)-...)
Affinity DataIC50: 4.30E+5nMAssay Description:Inhibition of Capra hircus (goat) brain DPP-3 using Arg-Arg-4mbetaNA as substrate assessed as liberation of 4mbetaNA from substrateMore data for this Ligand-Target Pair
In DepthDetails Article

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