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Report error Found 19 of ic50 data for polymerid = 50006496
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624590(CHEMBL5425605)
Affinity DataIC50: 390nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624591(CHEMBL5415008)
Affinity DataIC50: 700nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624589(CHEMBL5414585)
Affinity DataIC50: 750nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624588(CHEMBL5428173)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM11979(MgrA inhibitor, 1 | CHEMBL115145 | 5-[(3-carboxy-4...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of DNMT3A/3L (unknown origin) using poly(2'-deoxyinosinic-2'-deoxycytidylic acid) as substrate after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624592(CHEMBL5404240)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50430056(CHEMBL2336409 | SGI-1027)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50448484(CHEMBL3126646)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human DNMT3A2/3L using unmethylated DNA as substrate in presence of [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50430056(CHEMBL2336409 | SGI-1027)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DNMT3A2/3L using unmethylated DNA as substrate in presence of [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50448487(CHEMBL2385821)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human DNMT3A2/3L using unmethylated DNA as substrate in presence of [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50448489(CHEMBL3126651)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human DNMT3A2/3L using unmethylated DNA as substrate in presence of [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50448485(CHEMBL3126645)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of human DNMT3A2/3L using unmethylated DNA as substrate in presence of [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624588(CHEMBL5428173)
Affinity DataIC50: 6.47E+4nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3B (564 to 853 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624593(CHEMBL5415199)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624594(CHEMBL5406502)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3A (623 to 912 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624591(CHEMBL5415008)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3B (564 to 853 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624590(CHEMBL5425605)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3B (564 to 853 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624592(CHEMBL5404240)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3B (564 to 853 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed
TargetDNA (cytosine-5)-methyltransferase 3-like(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50624589(CHEMBL5414585)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition of N-terminal His-tagged human DNMT3B (564 to 853 residues)/N-terminal GST-tagged human DNMT3L (160 to 387 residues) co-expressed in bacul...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
PubMed