Compile Data Set for Download or QSAR
Report error Found 82 of ic50 data for polymerid = 50006386
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449597(CHEMBL4174825)
Affinity DataIC50: 238nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449561(CHEMBL4168457)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataIC50: 944nMAssay Description:Agonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as induction of beta-arrestin recruitment by measuring 2-(3-...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449598(CHEMBL4176317)
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449584(CHEMBL4169939)
Affinity DataIC50: 1.15E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449599(CHEMBL4169536)
Affinity DataIC50: 1.49E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449578(CHEMBL4159298)
Affinity DataIC50: 1.71E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449560(CHEMBL4168388)
Affinity DataIC50: 1.73E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449577(CHEMBL4162436)
Affinity DataIC50: 2.29E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449564(CHEMBL4171815)
Affinity DataIC50: 2.38E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449587(CHEMBL4161205)
Affinity DataIC50: 3.25E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449579(CHEMBL4172931)
Affinity DataIC50: 3.59E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449565(CHEMBL4177155)
Affinity DataIC50: 4.78E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449563(CHEMBL4161619)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataIC50: 5.99E+3nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398222(CHEMBL2177264)
Affinity DataIC50: 8.10E+3nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448075(CHEMBL1258979)
Affinity DataIC50: 9.91E+3nMAssay Description:Inverse agonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 7.5 uM THC-mediated beta-arrestin recruitment after 90 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449590(CHEMBL4160494)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449567(CHEMBL4176334)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449582(CHEMBL4170355)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449602(CHEMBL4166952)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449601(CHEMBL4173804)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449594(CHEMBL4159299)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398237(CHEMBL2177249)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398229(CHEMBL2177257)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449596(CHEMBL4163080)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449600(CHEMBL4159050)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449586(CHEMBL4171382)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449589(CHEMBL4173561)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449588(CHEMBL4169314)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561704(CHEMBL4793383)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448074(Emindole Sb)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 10 uM THC-mediated beta-arrestin recruitment after 90 mins by bet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221680(9-(2-(1H-indol-3-yl)ethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561707(CHEMBL4781871)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221704(9-(3,4-dimethoxyphenethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221703(9-(4-methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221681(9-(4-chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50221697(1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50212814(9-(4-chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449562(CHEMBL4165036)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561703(CHEMBL4745658)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561702(CHEMBL4755181)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561701(CHEMBL4755420)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50561700(CHEMBL1584113)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50552130(CHEMBL499876)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50056486(((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoylamino)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Prolink1-tagged human GPR18 receptor expressed in CHO cells assessed as inhibition of THC-induced beta arrestin recruitment af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50449595(CHEMBL4169940)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50434876(CHEMBL2387539)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50434881(CHEMBL2181545)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50398217(CHEMBL2181543)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 82 total ) | Next | Last >>
Jump to: