Compile Data Set for Download or QSAR
Report error Found 38 of ic50 data for polymerid = 50006371
LigandPNGBDBM50117663(CHEMBL3613707)
Affinity DataIC50: 6nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117662(CHEMBL3613706)
Affinity DataIC50: 6nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117663(CHEMBL3613707)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117662(CHEMBL3613706)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50433269(CHEMBL2376303)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50: 63nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50: 63nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50: 72nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50: 79nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50: 92nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50: 100nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50433274(CHEMBL2376321)
Affinity DataIC50: 126nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50: 204nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117665(CHEMBL3613709)
Affinity DataIC50: 205nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117666(CHEMBL3613710)
Affinity DataIC50: 365nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50: 389nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117668(CHEMBL3613712)
Affinity DataIC50: 394nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50433272(CHEMBL2376325)
Affinity DataIC50: 398nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117666(CHEMBL3613710)
Affinity DataIC50: 398nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117664(CHEMBL3613708)
Affinity DataIC50: 597nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117664(CHEMBL3613708)
Affinity DataIC50: 631nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117659(CHEMBL3613703)
Affinity DataIC50: 631nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117659(CHEMBL3613703)
Affinity DataIC50: 682nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50: 760nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117667(CHEMBL3613711)
Affinity DataIC50: 794nMAssay Description:Inhibition of human MGAT3 expressed in HEK293 cells assessed as effect on incorporation of [1,3-14C] glycerol into TAG by TLC method in presence of D...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM201239(US9187424, 6-2)
Affinity DataIC50: 820nMAssay Description:Inhibition of human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50579519(CHEMBL3912712)
Affinity DataIC50: 820nMAssay Description:Inhibition of human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50579526(CHEMBL4878564)
Affinity DataIC50: 820nMAssay Description:Inhibition of human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50117660(CHEMBL3613704)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50433273(CHEMBL2376322)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human recombinant MGAT3 expressed in insect cell membrane using 2-oleyl-sn-glycerol and [14C]-oleyl-coenzyme A as substrate after 10 to...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117660(CHEMBL3613704)
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117661(CHEMBL3613705)
Affinity DataIC50: 3.84E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117661(CHEMBL3613705)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM289003(US10093650, Example 16 | US10093650, Example 14 | ...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant human MGAT3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50090510(CHEMBL3581716)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibition of full length human MGAT3 transfected in Sf-21 cells using [1-14C]oleoyl-CoA assessed as incorporation of radioactivity into lip...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM276750(US10071992, Example 3.4 | (S)-2-(5-((3-ethoxypyrid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human MGAT3 using [1-14C]decanoyl-CoA and 1,2-didecanoyl-sn-glycerol as substrates assessed as incorporation of [1-14C]decanoyl into di...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM276748(US10071992, Example 3.5 | US10071992, Example 5 | ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human MGAT3 using [1-14C]decanoyl-CoA and 1,2-didecanoyl-sn-glycerol as substrates assessed as incorporation of [1-14C]decanoyl into di...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM504484(2-{5-[(3-Ethoxypyridin-2-yl)oxy]pyridin-3-yl}-N-[(...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of MGAT3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed