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TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645341(CHEMBL5563118)
Affinity DataIC50: 0.00200nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645339(CHEMBL5574302)
Affinity DataIC50: 0.0350nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645324(CHEMBL5576026)
Affinity DataIC50: 0.0840nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645320(CHEMBL5574055)
Affinity DataIC50: 0.155nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645342(CHEMBL5575835)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50587785(CHEMBL5178368)
Affinity DataIC50: 2nMAssay Description:Inhibition of haspin (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50587785(CHEMBL5178368)
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50587785(CHEMBL5178368)
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50605473(CHEMBL5186093)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50587785(CHEMBL5178368)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50603975(CHEMBL5201780)
Affinity DataIC50: 3nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645329(CHEMBL5563528)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50246769(CHEMBL4064608)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human haspin (471 end residues) expressed in baculovirus infected Sf21 insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50587785(CHEMBL5178368)
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681768(US20240199630, Compound 1)
Affinity DataIC50: 4.80nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50603974(CHEMBL5201904)
Affinity DataIC50: 5nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645340(CHEMBL5575484)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681770(US20240199630, Compound 2 | US20240199630, Compoun...)
Affinity DataIC50: 5.03nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 5.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681783(US20240199630, Compound 34)
Affinity DataIC50: 5.87nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681783(US20240199630, Compound 34)
Affinity DataIC50: 5.87nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50510133(CHEMBL4446681)
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681781(US20240199630, Compound 33)
Affinity DataIC50: 6.37nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681781(US20240199630, Compound 33)
Affinity DataIC50: 6.37nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50645335(CHEMBL5566424)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350270(US10208056, Compound 105)
Affinity DataIC50: 8.82nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350269(US10208056, Compound 104)
Affinity DataIC50: 8.91nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350253(US10208056, Compound 80)
Affinity DataIC50: 9.56nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350256(US10208056, Compound 83)
Affinity DataIC50: 9.80nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50442757(CHEMBL2443026)
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50442758(CHEMBL2443139)
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50442759(CHEMBL2443138)
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50442760(CHEMBL2443044)
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50407809(CHEMBL5095897)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50343559(1-(2-HYDROXYETHYL)-8-[[5-(4-METHYLPIPERAZIN-1-YL)-...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM681772(US20240199630, Compound 3 | US20240199630, Compoun...)
Affinity DataIC50: 10.2nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50603992(CHEMBL5179988)
Affinity DataIC50: 11nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50466167(CHEMBL4278808)
Affinity DataIC50: 12nMAssay Description:Inhibition of Haspin (unknown origin) after 3 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50605464(CHEMBL5188318)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350255(US10208056, Compound 82)
Affinity DataIC50: 12.8nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50542441(CHEMBL4642838)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50466167(CHEMBL4278808)
Affinity DataIC50: 14nMAssay Description:Inhibition of haspin (unknown origin) incubated for 3 hrs by ADP-GloTM kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50636431(CHEMBL5561973)
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50466167(CHEMBL4278808)
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350183(US10208056, Compound 15)
Affinity DataIC50: 15.9nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350264(US10208056, Compound 91)
Affinity DataIC50: 16.5nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM350266(US10208056, Compound 94)
Affinity DataIC50: 17.5nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2019
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human haspin using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human haspin using Histone H3 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
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