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TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50512854(CHEMBL4468747 | US11066363, Compound 37)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50500357(CHEMBL3746522 | US11066363, Compound 31)
Affinity DataIC50: 6.60nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50500359(CHEMBL3747611 | US11066363, Compound 13)
Affinity DataIC50: 7.46nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50500351(CHEMBL3746960 | US11066363, Compound 19)
Affinity DataIC50: 8.57nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50500356(CHEMBL3747406 | US11066363, Compound 7)
Affinity DataIC50: 12.4nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM504520(9-ethyl-6,6-dimethyl-11-oxo-8- (pyrimidin-5-yl)-6,...)
Affinity DataIC50: 12.5nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM504519((9-ethyl-6,6-dimethyl-11-oxo-8- (pyridin-4-yl)-6,1...)
Affinity DataIC50: 13.2nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50500353(CHEMBL3746395 | US11066363, Compound 10)
Affinity DataIC50: 14.5nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50500355(CHEMBL3747108 | US11066363, Compound 36)
Affinity DataIC50: 23.6nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50362781(CHEMBL1738797 | US9126931, 366 | Alectinib | 12565...)
Affinity DataIC50: 28.2nMAssay Description:SRPK1 Inhibitory Activities of the Compounds.More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617302(CHEMBL5085558)
Affinity DataIC50: 80nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50512854(CHEMBL4468747 | US11066363, Compound 37)
Affinity DataIC50: 98nMAssay Description:Inhibition of SRPK2 (unknown origin) incubated for 1 hr in presence of ATP by fluorescent plate reader methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617308(CHEMBL5397100)
Affinity DataIC50: 147nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617306(CHEMBL5435975)
Affinity DataIC50: 147nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 185nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50564378(CHEMBL4787157)
Affinity DataIC50: 203nMAssay Description:Inhibition of SRPK2 (unknown origin) incubated for 10 mins in presence of ATP by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617313(CHEMBL5405335)
Affinity DataIC50: 210nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 227nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM221074(US9695160, 12 | SPHINX31 | US9796707, Compound 12)
Affinity DataIC50: 256nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617299(CHEMBL5439515)
Affinity DataIC50: 260nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617311(CHEMBL5416930)
Affinity DataIC50: 300nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617312(CHEMBL5437009)
Affinity DataIC50: 340nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617310(CHEMBL5409896)
Affinity DataIC50: 460nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617297(CHEMBL5407046)
Affinity DataIC50: 510nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617307(CHEMBL5409387)
Affinity DataIC50: 626nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617300(CHEMBL5398076)
Affinity DataIC50: 660nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617298(CHEMBL5399262)
Affinity DataIC50: 670nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617294(CHEMBL5433267)
Affinity DataIC50: 750nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617296(CHEMBL5422948)
Affinity DataIC50: 870nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617305(CHEMBL5403164)
Affinity DataIC50: 900nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617301(CHEMBL5416263)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50235034(CHEMBL4064277)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617292(CHEMBL5434661)
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617293(CHEMBL5416898)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617295(CHEMBL5415454)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617291(CHEMBL5417678)
Affinity DataIC50: 3.77E+3nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50235034(CHEMBL4064277)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of SRPK2 (unknown origin) incubated for 10 mins in presence of ATP by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SRPK2 using [GRSRSRSRSR] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human SRPK2 (46 to end residues) using RSRSRSRSRSRSRSR as substrate incubated for 40 mins in presence of [gamma33P]ATP by r...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617309(CHEMBL5085599)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617304(CHEMBL5421441)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617303(CHEMBL5409358)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50617290(CHEMBL5410156)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human SRPK2 using GRSRSRSRSR as substrate in presence of [gamma-33p]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human GST-tagged SRPK2 expressed in baculovirus expression system using serine/threonine-07 peptide as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed