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TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612791(CHEMBL5280560)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50503137(CHEMBL4516990)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of wild type GST-tagged ULK1 (unknown origin) after 5 mins in presence of gamma-[32]P-ATP by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612793(CHEMBL5266681)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379404(6-((4-(cyclopropylamino)-5-(trifluoromethyl)pyrimi...)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379381(N4-cyclopropyl-N2-(quinolin-6-yl)-5-(trifluorometh...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379329(N2-(1H-benzo[d]imidazol-6-yl)-N4-cyclopropyl-5-(tr...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379305(N2-(1H-benzo[d][1,2,3]triazol-6-yl)-N4-cyclopropyl...)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379307(N4-cyclopropyl-N2-(3,4-dihydro-2H-benzo[b][1,4]dio...)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal SUMO-tagged ULK1 kinase domain (1 to 283 residues) (unknown origin) using MBP as substrate in presence of [32P]ATP after 15 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 8nMAssay Description:Inhibition of ULK1 (unknown origin) by 32P-ATP radio active assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 8nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612792(CHEMBL5269042)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50520142(CHEMBL4435393)
Affinity DataIC50: 9nMAssay Description:Inhibition of wild-type human partial length ULK1 (M1 to T309 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human ULK1 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 10.3nMAssay Description:Inhibition of human ULK1 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50280086(CHEMBL4167070)
Affinity DataIC50: 11nMAssay Description:Inhibition of ATG13 binding to full-length ULK1 (unknown origin) expressed in HEK293T cells preincubated for 15 mins followed by human C-terminal FLA...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379450(US10266549, Example 349 | US10774092, Example 349)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379414(N-(4-((4-(cyclopropylamino)-5-(trifluoromethyl)pyr...)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379408(N4-cyclopropyl-N2-(quinoxalin-6-yl)-5-(trifluorome...)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379352(N4-cyclopropyl-N2-(5-methoxypyridin-3-yl)-5-(trifl...)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379311(N4-cyclopropyl-N2-(1H-indazol-5-yl)-5-(trifluorome...)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379259(US10266549, Example 158a | US10774092, Example 158...)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379387(N4-cyclopropyl-N2-(quinolin-3-yl)-5-(trifluorometh...)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379264(US10266549, Example 161a | US10774092, Example 161...)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379325(US10266549, Example 208a | US10774092, Example 208...)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379406(US10266549, Example 304a | US10774092, Example 304...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379332(N2-(benzo[d][1,3]dioxol-5-yl)-N4-cyclopropyl-5-(tr...)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379323(N4-cyclopropyl-N2-(1H-indol-5-yl)-5-(trifluorometh...)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50280041(CHEMBL4159827)
Affinity DataIC50: 24nMAssay Description:Inhibition of ATG13 binding to full-length ULK1 (unknown origin) expressed in HEK293T cells preincubated for 15 mins followed by human C-terminal FLA...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50520161(CHEMBL4468020 | US10894784, Example 39.01.02)
Affinity DataIC50: 28nMAssay Description:Inhibition of wild-type human partial length ULK1 (M1 to T309 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379252(US10266549, Example 152a | US10774092, Example 152...)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379413(N-(cyclopropanecarbonyl)-N-(4-((4-(cyclopropylamin...)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379445(N4-cyclopropyl-N2-(4-ethyl-3,4-dihydro-2H-pyrido[3...)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612787(CHEMBL5279228)
Affinity DataIC50: 31nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612790(CHEMBL5276694)
Affinity DataIC50: 31nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379295(US10266549, Example 182a | US10774092, Example 182...)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50280098(CHEMBL4176003)
Affinity DataIC50: 40nMAssay Description:Inhibition of ATG13 binding to full-length ULK1 (unknown origin) expressed in HEK293T cells preincubated for 15 mins followed by human C-terminal FLA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379343(US10266549, Example 221a | US10774092, Example 221...)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379376(N4-cyclopropyl-N2-(2,2-difluorobenzo[d][1,3]dioxol...)
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50271370(CHEMBL4127042)
Affinity DataIC50: 45nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50280093(CHEMBL4170480)
Affinity DataIC50: 45nMAssay Description:Inhibition of ATG13 binding to full-length ULK1 (unknown origin) expressed in HEK293T cells preincubated for 15 mins followed by human C-terminal FLA...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50: 45nMAssay Description:Inhibition of wild type GST-tagged ULK1 (unknown origin) after 5 mins in presence of gamma-[32]P-ATP by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50556418(CHEMBL4784530)
Affinity DataIC50: 45nMAssay Description:Inhibition of ULK1 (unknown origin) by 32P-ATP radio active assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612794(CHEMBL5288376)
Affinity DataIC50: 45nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379374(2-((4-(cyclopropylamino)-5-(trifluoromethyl)pyrimi...)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111575(CHEMBL3603853)
Affinity DataIC50: 67nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM17051(N-{3-[(5-iodo-4-{[3-(thiophen-2-ylformamido)propyl...)
Affinity DataIC50: 87nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379177(US10266549, Example 88 | US10266549, Example 171a ...)
Affinity DataIC50: 108nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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