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TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612791(CHEMBL5280560)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50637636(CHEMBL5568152)
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50637636(CHEMBL5568152)
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111572(CHEMBL3605057)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of GST-tagged ULK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50503137(CHEMBL4516990)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of wild type GST-tagged ULK1 (unknown origin) after 5 mins in presence of gamma-[32]P-ATP by immunoblot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612793(CHEMBL5266681)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50503137(CHEMBL4516990)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50503137(CHEMBL4516990)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379404(6-((4-(cyclopropylamino)-5-(trifluoromethyl)pyrimi...)
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379381(N4-cyclopropyl-N2-(quinolin-6-yl)-5-(trifluorometh...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379329(N2-(1H-benzo[d]imidazol-6-yl)-N4-cyclopropyl-5-(tr...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of SUMO-tagged ULK1 (unknown origin) kinase domain expressed in KRX cells using [32P]-gamma-ATP and myelin basic protein substrate incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379305(N2-(1H-benzo[d][1,2,3]triazol-6-yl)-N4-cyclopropyl...)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM379307(N4-cyclopropyl-N2-(3,4-dihydro-2H-benzo[b][1,4]dio...)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human ULK1 (1-649) expressed in Sf9 cells using myelin basic protein as substrate by ADP-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal SUMO-tagged ULK1 kinase domain (1 to 283 residues) (unknown origin) using MBP as substrate in presence of [32P]ATP after 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 8nMAssay Description:Inhibition of ULK1 (unknown origin) by 32P-ATP radio active assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
Affinity DataIC50: 8nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50111577(CHEMBL3605055)
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50612792(CHEMBL5269042)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of ULK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50637406(CHEMBL4744680)
Affinity DataIC50: 8.30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50637406(CHEMBL4744680)
Affinity DataIC50: 8.30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50637406(CHEMBL4744680)
Affinity DataIC50: 8.30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50520142(CHEMBL4435393)
Affinity DataIC50: 9nMAssay Description:Inhibition of wild-type human partial length ULK1 (M1 to T309 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human ULK1 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 9.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737767(5-(2-((7-chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737769(5-(2-((7-chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737770(2-(2-((7-chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737771(5-(2-((2-(azetidin-3-yl)-7-chloro- 1,2,3,4-tetrahy...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737773(5-(2-((6-chloroisoindolin-5- yl)amino)-5- (trifluo...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737775(5-(2-((7-ethyl-1,2,3,4- tetrahydroisoquinolin-6-yl...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737776(5-(2-((7-cyclopropyl-1,2,3,4- tetrahydroisoquinoli...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737778(5-(2-((6-chloro-2-(1- methylazetidin-3-yl)isoindol...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737779(5-(2-((7-ethyl-2-methyl-1,2,3,4- tetrahydroisoquin...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737780(5-(2-((7-cyclopropyl-2-methyl- 1,2,3,4-tetrahydroi...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737782(N-(5-(2-((7-chloro-1,2,3,4- tetrahydroisoquinolin-...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737783(5-(2-((6-Chloro-2- methylisoindolin-5-yl)amino)-5-...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737785(5-(2-((6-Cyclopropyl-2- methylisoindolin-5-yl)amin...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737787(2-(2-((7-Chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737789(2-(2-((7-chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737790(2-(2-((7-Chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737794(5-(2-((7-Chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737795(2-(2-((7-Chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737796(2-(2-((7-Cyclopropyl-1,2,3,4- tetrahydroisoquinoli...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737797(2-(2-((7-Chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737798(2-(2-((7-Chloro-1,2,3,4- tetrahydroisoquinolin-6-y...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737799(7-Chloro-N-(4-(4- (methylsulfonyl)thiophen-2-yl)-5...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737800(2-(2-((6-Chloroisoindolin-5- yl)amino)-5- (trifluo...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737801(2-(2-((7-ethyl-1,2,3,4- tetrahydroisoquinolin-6-yl...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase ULK1(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM737802(2-(2-((7-(Methylthio)-1,2,3,4- tetrahydroisoquinol...)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

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