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TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of DAPK1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50536679(CHEMBL4568087)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of human DAPK1 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human DAPK1 using KKLNRTLSFAEPG as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50536678(CHEMBL4550702)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50536675(CHEMBL4569508)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50499279(CHEMBL3735890)
Affinity DataIC50: 12nMAssay Description:Inhibition of DAPK1 (unknown origin) by electrophoretic mobility shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 13nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 13.1nMAssay Description:Inhibition of human DAPK1 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 13.1nMAssay Description:Inhibition of human DAPK1 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 15.7nMAssay Description:Inhibition of human DAPK1 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50554817(CHEMBL4764610)
Affinity DataIC50: 23nMAssay Description:Inhibition of human DAPK1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50536681(CHEMBL4552628)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human GST-tagged DAPK1 catalytic domain expressed in baculovirus expression system by Adapta assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50166251(CHEMBL3799389)
Affinity DataIC50: 140nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataIC50: 200nMAssay Description:Inhibition of DAPK1 (unknown origin) by (33P-ATP) filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM104065(HS38)
Affinity DataIC50: 200nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50506351(CHEMBL4439133)
Affinity DataIC50: 203nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged DAPK1 catalytic domain (1 to 363 residues) expressed in baculovirus expression system by Adapta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50616759(CHEMBL5407750)
Affinity DataIC50: 247nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 247nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50616760(CHEMBL5433785)
Affinity DataIC50: 370nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50166254(CHEMBL3797466)
Affinity DataIC50: 450nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50166076(CHEMBL3799585)
Affinity DataIC50: 510nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM311261(US10155760, Example 117 | (S)-methyl (5-((2-amino-...)
Affinity DataIC50: 560nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50166077(CHEMBL513703)
Affinity DataIC50: 700nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM311210(US10155760, Example 66 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 810nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM67454(MLS002473304 | purpurin | 1,2,4-tris(oxidanyl)anth...)
Affinity DataIC50: 890nMAssay Description:Inhibition of DAPK1 (1 to 285 residues) (unknown origin) expressed in Escherichia coli using KKLNRTLSFAEPG as substrate in presence of ATP by fluoro-...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520846(CHEMBL4461911)
Affinity DataIC50: 920nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 100 uM [gamma-33P]-ATP by filtration met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50462709(CHEMBL4245507)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520846(CHEMBL4461911)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50121391(CHEMBL3622137)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant DAPK1 (unknown origin) using fluoresceinated peptide as substrate after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM311208(US10155760, Example 64 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM26658(2-(2,4-dihydroxyphenyl)-3,5,7-trihydroxychromen-4-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of ANS from DAPK1 catalytic domain (1 to 285) (unknown origin) after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50166121(CHEMBL3797480)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50616763(CHEMBL5412508)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of DAPK1 (unknown origin) in presence of 33P-ATP radiolabeled kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520847(CHEMBL4467582)
Affinity DataIC50: 2.61E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520849(CHEMBL4461940)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520848(CHEMBL4464585)
Affinity DataIC50: 2.77E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520846(CHEMBL4461911)
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 1 uM [gamma-33P]-ATP by filtration metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50206434(1,2-dihydroxyanthracene-9,10-dione | alizarin | 1,...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of DAPK1 (1 to 285 residues) (unknown origin) expressed in Escherichia coli using KKLNRTLSFAEPG as substrate in presence of ATP by fluoro-...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520854(CHEMBL4521651)
Affinity DataIC50: 4.29E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520846(CHEMBL4461911)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of DAPK1 in HEK293 tau-BiFC cells assessed as reduction in forskolin-induced tau aggregation after 48 hrs by Hoechst staining based HCS an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50616762(CHEMBL5426378)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of DAPK1 (unknown origin) in presence of 33P-ATP radiolabeled kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50520852(CHEMBL4568513)
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 8.90E+3nMAssay Description:Displacement of ANS from DAPK1 catalytic domain (1 to 285) (unknown origin) after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50552171(CHEMBL4757567)
Affinity DataIC50: 8.95E+3nMAssay Description:Inhibition of human DAPK1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50616764(CHEMBL5028838)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of DAPK1 (1 to 285 residues) (unknown origin) expressed in Escherichia coli using KKLNRTLSFAEPG as substrate in presence of ATP by fluoro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DAPK1 using [KKLNRTLSFAEPG] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50166260(CHEMBL3799505)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DAPK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50208911(CHEMBL3884319)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged DAPK1 catalytic domain (1 to 363 residues) expressed in baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDeath-associated protein kinase 1(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM7462(cid_5280863 | CHEMBL150 | 3,5,7-trihydroxy-2-(4-hy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of ANS from DAPK1 catalytic domain (1 to 285) (unknown origin) after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
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