Compile Data Set for Download or QSAR
Report error Found 32 of ic50 data for polymerid = 50000996
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50: 8nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525914(CHEMBL4558285)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM113069(US9695194, 5)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human KLK14 using S-2302 substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525895(CHEMBL4447752)
Affinity DataIC50: 126nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525904(CHEMBL4461533)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525905(CHEMBL4517343)
Affinity DataIC50: 251nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525912(CHEMBL4543039)
Affinity DataIC50: 316nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525899(CHEMBL4465265)
Affinity DataIC50: 398nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525900(CHEMBL4460168)
Affinity DataIC50: 398nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525917(CHEMBL4579813)
Affinity DataIC50: 794nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM51911(3-(2-methoxyphenyl)-3-(4-methoxyphenyl)-N-[(4-prop...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM32709(1-(4-methylbenzoyl)-3-(3-pyridinyl)-1H-1,2,4-triaz...)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525911(CHEMBL4535907)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525903(CHEMBL4436048)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM33453((3-Amino-[1,2,4]triazol-4-yl)-(4-methoxy-phenyl)-m...)
Affinity DataIC50: 3.43E+3nMAssay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50522493(CHEMBL4530083)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of recombinant C-terminal 10His-tagged human KLK14 (Gln19 to Met248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525918(CHEMBL4473069)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525913(CHEMBL4464120)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525897(CHEMBL4536142)
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM33882(SMR000306508 | (5-azanyl-3-pyridin-3-yl-1,2,4-tria...)
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM33437(MLS000099650 | SMR000074479 | 1-(3,4-dimethoxybenz...)
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525901(CHEMBL4448315)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50525902(CHEMBL4547455)
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444599(CHEMBL3099875)
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444600(CHEMBL1462676)
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)
Affinity DataIC50: 9.90E+4nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)
Affinity DataIC50: 1.12E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKallikrein-14(Human)
German Cancer Research Center (Dkfz)

Curated by ChEMBL
LigandPNGBDBM50444596(CHEMBL3099883)
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed