Compile Data Set for Download or QSAR
Report error Found 27 of ic50 data for polymerid = 50000507
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259563(2-{[3,4-Dioxo-2-(pyridin-4-ylamino)cyclobut-1-en-1...)
Affinity DataIC50: 160nMAssay Description:Inhibition of CK1-gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259376(3-{[(1R)-1-phenylethyl]amino}-4-(pyridin-4-ylamino...)
Affinity DataIC50: 250nMAssay Description:Inhibition of CK1-gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259532(2-{[3,4-Dioxo-2-(pyridin-4-ylamino)cyclobut-1-en-1...)
Affinity DataIC50: 520nMAssay Description:Inhibition of CK1-gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259637(3-{[2-(2-Furyl)pyridin-4-yl]amino}-4-{[(1R)-1-phen...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of CK1-gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)
Affinity DataIC50: 5.52E+3nMAssay Description:Inhibition of CK1gamma1 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 7.17E+3nMAssay Description:Inhibition of human CK1gamma1 using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of human CK1gamma1 using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50311985(3-(7-(4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]h...)
Affinity DataIC50: 9.51E+3nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50401152(CHEMBL2205766)
Affinity DataIC50: 9.55E+3nMAssay Description:Inhibition of CSNK1G1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CK1gamma1(25 to 355 residues) using KRRRALS(p)VAS as substrate incubated for 40 mins in presence of [gamma-33ATP] by ...More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CK1gamma1 using [KRRRAL[pS]VASLPGL] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50499634(CHEMBL3741589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CK1gamma1 (unknown origin)More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50357884(CHEMBL1916359)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259638(3-{[2-(3-Thienyl)pyridin-4-yl]amino}-4-{[(1R)-1-ph...)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of CK1-gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316252(methyl 4-(6-(4-aminophenyl)-4-morpholino-1H-pyrazo...)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50094893(cid_8323 | CHEMBL88326 | 1-hydroxy-4-amino-anthraq...)
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diaminoanthracene-9,10-dione | 1,4-diamino-ant...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-dihydroxyanthracene-9,10-dione | quinizarin | ...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316253(tert-Butyl 4-(6-(4-aminophenyl)-4-morpholino-1H-py...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50311953(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-methylpipe...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50259601(3-{[2-(2-Fluorophenyl)pyridin-4-yl]amino}-4-{[(1R)...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1-gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50378568(CHEMBL1163016)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50311954(6-methyl-4-(4-methyl-1H-indol-5-ylamino)-5-(3-(4-m...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50315069(1-(4-(4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-6-(t...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human full-length GST-tagged CSNK1G1 expressed in baculovirus expression system using FRET-labeled Ser/Thr 05 peptide as su...More data for this Ligand-Target Pair
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PubMed