Compile Data Set for Download or QSAR
Report error Found 87 of ic50 data for polymerid = 50000266,50002275
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 0.130nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50276748([(1R,3S,9S,11S,14R)-9-(3-Guanidino-propyl)-4,7,10,...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277112(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50: 1nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277111(3-Benzo[1,3]dioxol-5-yl-3-[1-oxo-6-(1,2,3,4-tetrah...)
Affinity DataIC50: 2nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Mouse)
University of Bradford

Curated by ChEMBL
LigandPNGBDBM50083811(3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at mouse endothelial alphavbeta3 integrin receptor by cell adhesion assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277112(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50: 5nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50276748([(1R,3S,9S,11S,14R)-9-(3-Guanidino-propyl)-4,7,10,...)
Affinity DataIC50: 5.64nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277098(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50: 7nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296598((R)-2-(2,4-dichlorophenylsulfonamido)-3-(thiophene...)
Affinity DataIC50: 8nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50265535(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 10.8nMAssay Description:Displacement of [125I]c(RGDyK) form integrin alphaVbeta3 receptor in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296610((R)-3-(1-methyl-1H-pyrazole-5-carboxamido)-2-(2,4,...)
Affinity DataIC50: 11nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50265534(2-((2R,8R,11R,14S)-11-(4-aminobutyl)-8-(3-guanidin...)
Affinity DataIC50: 11.2nMAssay Description:Displacement of [125I]c(RGDyK) form integrin alphaVbeta3 receptor in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50265536(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 13.8nMAssay Description:Displacement of [125I]c(RGDyK) form integrin alphaVbeta3 receptor in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277111(3-Benzo[1,3]dioxol-5-yl-3-[1-oxo-6-(1,2,3,4-tetrah...)
Affinity DataIC50: 14nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50276746(c[RGDf-(3S)-Carboxymorpholine] | CHEMBL452724)
Affinity DataIC50: 15.1nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 18.9nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296635((R)-2-(2,3-dichlorophenylsulfonamido)-3-(thiophene...)
Affinity DataIC50: 19nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50276747(c[RGDf-(3R)-Carboxymorpholine] | CHEMBL443362)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta5 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296597((R)-3-(thiophene-3-carboxamido)-2-(2,4,6-trichloro...)
Affinity DataIC50: 24nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296603((R)-3-benzamido-2-(2-iodophenylsulfonamido)propano...)
Affinity DataIC50: 25nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296611((R)-3-(furan-3-carboxamido)-2-(2,4,6-trimethylphen...)
Affinity DataIC50: 32nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50276747(c[RGDf-(3R)-Carboxymorpholine] | CHEMBL443362)
Affinity DataIC50: 32.6nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277096(3-(6-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: 39nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296609((R)-3-(2-methyloxazole-4-carboxamido)-2-(2,4,6-tri...)
Affinity DataIC50: 41nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296612((R)-3-(thiophene-3-carboxamido)-2-(2,4,6-trimethyl...)
Affinity DataIC50: 44nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296600((R)-3-benzamido-2-(2,3-dichlorophenylsulfonamido)p...)
Affinity DataIC50: 62nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296607((R)-3-(pyrimidine-5-carboxamido)-2-(2,4,6-trimethy...)
Affinity DataIC50: 63nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50265536(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 73.3nMAssay Description:Displacement of [125I][Tyr4]BBN form integrin alphaVbeta3 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296632((R)-3-(2-methoxybenzamido)-2-(2,4,6-trimethylpheny...)
Affinity DataIC50: 78nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50265537((S)-N1-((5R,8S,11R,17R,20S,23R)-11-((1H-imidazol-4...)
Affinity DataIC50: 79.0nMAssay Description:Displacement of [125I][Tyr4]BBN form integrin alphaVbeta3 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296608((R)-3-(nicotinamido)-2-(2,4,6-trimethylphenylsulfo...)
Affinity DataIC50: 81nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50265535(2-((2R,8R,11R,14S)-11-((5R,8S,11R,17R,20S,23R,26S)...)
Affinity DataIC50: 85.5nMAssay Description:Displacement of [125I][Tyr4]BBN form integrin alphaVbeta3 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296596((R)-2-(3-cyanophenylsulfonamido)-3-(furan-3-carbox...)
Affinity DataIC50: 98nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296599((R)-3-benzamido-2-(2,6-dichlorophenylsulfonamido)p...)
Affinity DataIC50: 118nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296623((R)-3-benzamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50: 120nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50276746(c[RGDf-(3S)-Carboxymorpholine] | CHEMBL452724)
Affinity DataIC50: 157nMAssay Description:Displacement of [125I]echistatin from integrin alphaVbeta3 receptor in human placenta by microplate scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277095(3-(5-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: 180nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296595((R)-3-(furan-3-carboxamido)-2-(3-methoxyphenylsulf...)
Affinity DataIC50: 208nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277075(3-(4-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: 230nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296604((R)-3-benzamido-2-(2-chlorophenylsulfonamido)propa...)
Affinity DataIC50: 260nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296633((R)-3-(furan-3-carboxamido)-2-(2-methylphenylsulfo...)
Affinity DataIC50: 260nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296606((R)-3-(isonicotinamido)-2-(2,4,6-trimethylphenylsu...)
Affinity DataIC50: 301nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277098(3-[1-Oxo-6-(1,2,3,4-tetrahydro-benzo[4,5]imidazo[1...)
Affinity DataIC50: 310nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296605((R)-3-benzamido-2-(2-methylphenylsulfonamido)propa...)
Affinity DataIC50: 320nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277097(3-(7-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: 370nMAssay Description:Binding affinity to human integrin alphavbeta3 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50277096(3-(6-(2-amino-1-methyl-1H-benzo[d]imidazol-4-yloxy...)
Affinity DataIC50: 600nMAssay Description:Binding affinity to human integrin alphavbeta5 receptor by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296634((R)-3-(furan-3-carboxamido)-2-(2-methoxyphenylsulf...)
Affinity DataIC50: 700nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296601((R)-3-benzamido-2-(2-methoxyphenylsulfonamido)prop...)
Affinity DataIC50: 729nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296594((R)-3-(furan-3-carboxamido)-2-(pyridine-3-sulfonam...)
Affinity DataIC50: 793nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrin alpha-V(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50296629((R)-3-acetamido-2-(2,4,6-trimethylphenylsulfonamid...)
Affinity DataIC50: 800nMAssay Description:Inhibition of fibrinogen binding to alphavbeta3 integrinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 87 total ) | Next | Last >>
Jump to: