Compile Data Set for Download or QSAR
Report error Found 344 of ic50 data for polymerid = 49001069,49001070,50003864,50006370
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445384(CHEMBL3104469)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445385(CHEMBL3104468)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445368(CHEMBL3104466)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445378(CHEMBL3104642)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445386(CHEMBL3104641)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445384(CHEMBL3104469)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445385(CHEMBL3104468)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445368(CHEMBL3104466)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445378(CHEMBL3104642)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445386(CHEMBL3104641)
Affinity DataIC50: 0nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50558696(CHEMBL4777970)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302257((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-ethylpipera...)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302270((R)-2-(4-(6-chloropyrazin-2-ylamino)-1-(3,4-dimeth...)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302264((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-isopropylpi...)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50558695(CHEMBL4741230)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50543457(CHEMBL4635039)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302258((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-isopropylpi...)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50543458(CHEMBL4642307)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302250((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-isopropylpi...)
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50302272(ACT-058362 | CHEMBL1164032 | CHEMBL567303 | 1-(2-(...)
Affinity DataIC50: 3.60nMAssay Description:Binding affinity to human urotensin 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50252659((S)-N-(1-(3-bromo-4-(piperidin-4-yloxy)benzyl)pyrr...)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of urotensin 2-induced calcium mobiliz...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302266((R)-N-(4-(4-(4-cyclobutylpiperazin-1-yl)-1-oxoisoi...)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302271((R)-2-(1-(3,4-dimethoxyphenyl)-4-(6-methoxypyrazin...)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50459265(CHEMBL4205274)
Affinity DataIC50: 4nMAssay Description:Displacement of [Na125I]-synthetic URP from human UT receptor expressed in HEK293 cell membranes incubated for 2 hrs by gamma-countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302249((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-ethylpipera...)
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445383(CHEMBL3104471)
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50459261(CHEMBL4208184)
Affinity DataIC50: 5.40nMAssay Description:Displacement of [Na125I]-synthetic URP from human UT receptor expressed in HEK293 cell membranes incubated for 2 hrs by gamma-countingMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50459266(CHEMBL4217514)
Affinity DataIC50: 5.60nMAssay Description:Displacement of [Na125I]-synthetic URP from human UT receptor expressed in HEK293 cell membranes incubated for 2 hrs by gamma-countingMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302260((R)-2-(1-(3,4-dimethoxyphenyl)-4-(thiophen-2-ylmet...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302268(N-((R)-4-(3,4-dimethoxyphenyl)-4-(1-oxo-4-(4-((R)-...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50249878(SB-706375 | (R)-2-bromo-4,5-dimethoxy-N-(3-(1-meth...)
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]-U2 from human recombinant urotensin2 receptor expressed in human Chem-2 cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50508365(CHEMBL4457118)
Affinity DataIC50: 6nMAssay Description:Displacement of Eu-labelled UT2 from recombinant human UT2 receptor expressed in HEK293 cell membranes preincubated for 10 mins followed by Eu-labell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302259((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-ethylpipera...)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302261((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-ethylpipera...)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50543461(CHEMBL4638346)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50302257((R)-N-(4-(3,4-dimethoxyphenyl)-4-(4-(4-ethylpipera...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at urotensin 2 receptor in human RMS13 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobilization aft...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50249878(SB-706375 | (R)-2-bromo-4,5-dimethoxy-N-(3-(1-meth...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at urotensin 2 receptor in human RMS13 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobilization aft...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445376(CHEMBL3104644)
Affinity DataIC50: 8.90nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445376(CHEMBL3104644)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50508375(CHEMBL4525919)
Affinity DataIC50: 9nMAssay Description:Displacement of Eu-labelled UT2 from recombinant human UT2 receptor expressed in HEK293 cell membranes preincubated for 10 mins followed by Eu-labell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50224715(tert-butyl 4-(2-(5-chloro-2-(1-(2-(3-oxo-2,3-dihyd...)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat UT receptor transfected in CHOK1 cells assessed as calcium mobilization by FLIPR methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445370(CHEMBL3104464)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445370(CHEMBL3104464)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302252(N-((R)-4-(3,4-dimethoxyphenyl)-4-(1,3-dioxo-4-(4-(...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302253(N-((R)-4-(3,4-dimethoxyphenyl)-4-(1,3-dioxo-4-(4-(...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302254(N-((R)-4-(3,4-dimethoxyphenyl)-4-(1,3-dioxo-4-(4-(...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50445383(CHEMBL3104471)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50543459(CHEMBL4643905)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Human)
Laval University

Curated by ChEMBL
LigandPNGBDBM50036148(CHEMBL3358687)
Affinity DataIC50: 13nMAssay Description:Displacement of europium-labeled urotensin-II from human urotensin-2 receptor expressed in HEK293 cells by TRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrotensin-2 receptor(Rat)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50302265((R)-N-(4-(4-(4-cyclopropylpiperazin-1-yl)-1-oxoiso...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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