Compile Data Set for Download or QSAR
Report error Found 480 of ic50 data for polymerid = 49000639,50001604
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(ORG-25543 | 4-Benzyloxy-N-(1-dimethylamino-cyclope...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023929(CHEMBL3325502)
Affinity DataIC50: 15nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(ORG-25543 | 4-Benzyloxy-N-(1-dimethylamino-cyclope...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(ORG-25543 | 4-Benzyloxy-N-(1-dimethylamino-cyclope...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human GlyT-2 expressed in CHO cells assessed as reduction in [3H]-glycine uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(ORG-25543 | 4-Benzyloxy-N-(1-dimethylamino-cyclope...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human GlyT2 stably expressed in CHO cells assessed as reduction in [3H]glycine uptake incubated for 10 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(ORG-25543 | 4-Benzyloxy-N-(1-dimethylamino-cyclope...)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human GlyT2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138590(2-(7-Hydroxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537022(CHEMBL4587165)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human GlyT2 expressed in porcine aorta epithelial cells assessed as reduction in [3H]-Glycine uptake at pH 7.5 by scintillation spectro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537040(CHEMBL4515597)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138578(2-(7-Hydroxy-1-methyl-3,4-dihydro-1H-isoquinolin-2...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50203568((1-(4-(6-((5-(2-fluorophenyl)-1,2,4-oxadiazol-3-yl...)
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]glycine uptake at human GlyT2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537034(CHEMBL4572247)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138594(2-(5-Hydroxy-1,3-dihydro-isoindol-2-ylmethyl)-N-(4...)
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138558(2-[(6-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-ylam...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537044(CHEMBL4562565)
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537033(CHEMBL4535356)
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023797(CHEMBL3325511)
Affinity DataIC50: 52nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537043(CHEMBL4227139)
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138584(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-((E...)
Affinity DataIC50: 56nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138559(2-(7-Hydroxy-1,2,4,5-tetrahydro-benzo[d]azepin-3-y...)
Affinity DataIC50: 58nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023926(CHEMBL3325505)
Affinity DataIC50: 62nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537049(CHEMBL4527071)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023866(CHEMBL3325509)
Affinity DataIC50: 66nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138556(2-(7-Hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-2...)
Affinity DataIC50: 67nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537023(CHEMBL4542099)
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023928(CHEMBL3325503)
Affinity DataIC50: 71nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138565(N-[4-(4-Chloro-phenyl)-butyl]-2-{[2-(4-hydroxy-phe...)
Affinity DataIC50: 77nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102687(4-Butoxy-N-(1-dimethylamino-cyclopentylmethyl)-3,5...)
Affinity DataIC50: 77nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023930(CHEMBL3325501)
Affinity DataIC50: 80nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138555(2-[(6-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-ylam...)
Affinity DataIC50: 81nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50102688(4-Benzyloxy-N-(1-dimethylamino-cyclohexylmethyl)-3...)
Affinity DataIC50: 84nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138561(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 86nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138569(2-(7-Hydroxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl...)
Affinity DataIC50: 89nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50537054(CHEMBL4549008)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138572(N-[4-(3-Chloro-phenyl)-butyl]-2-{[2-(4-hydroxy-phe...)
Affinity DataIC50: 99nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023874(CHEMBL3325508)
Affinity DataIC50: 99nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human GlyT-2 expressed in HEK293 cells assessed as reduction in [3H]-glycine uptake preincubated for 30 mins followed by 3H]-glycine ad...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)
Affinity DataIC50: 100nMAssay Description:Inhibition of full length human GlyT2 expressed in FreeStyle 293-F suspension cells incubated for 30 mins before [3H]glycine addition and measured af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023924(CHEMBL3325507)
Affinity DataIC50: 105nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023924(CHEMBL3325507)
Affinity DataIC50: 105nMAssay Description:Inhibition of human GlyT-2 expressed in HEK293 cells assessed as reduction in [3H]-glycine uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023924(CHEMBL3325507)
Affinity DataIC50: 105nMAssay Description:Reversible inhibition of recombinant human GlyT2 expressed in HEK293 cells assessed as reduction in [3H]-glycine uptake after 2 hrs by top count assa...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023925(CHEMBL3325506)
Affinity DataIC50: 107nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50335008(5-Biphenyl-4-yl-4-(2-fluorophenyl)-N-methyl-4H-1,2...)
Affinity DataIC50: 110nMAssay Description:Inhibition of [3H]glycine uptake at GlyT2 in rat C6 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023993(CHEMBL3325495)
Affinity DataIC50: 112nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50023932(CHEMBL3325499)
Affinity DataIC50: 115nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138587(N-[4-(3,4-Dichloro-phenyl)-butyl]-2-{[2-(4-hydroxy...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138592(2-(6-Hydroxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138576(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-[4-...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50138575(2-[(2-Hydroxy-6,7,8,9-tetrahydro-5H-benzocyclohept...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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