Compile Data Set for Download or QSAR
Report error Found 63 of ic50 data for polymerid = 49000526,50000019,50000150,50000462,50002350
LigandPNGBDBM50488134(CHEMBL2283229)
Affinity DataIC50: 73nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488117(CHEMBL2283230)
Affinity DataIC50: 91nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488133(CHEMBL2283231)
Affinity DataIC50: 110nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488132(CHEMBL2283321)
Affinity DataIC50: 130nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488131(CHEMBL2283322)
Affinity DataIC50: 140nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488142(CHEMBL2283232)
Affinity DataIC50: 150nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488139(CHEMBL2283323)
Affinity DataIC50: 200nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488140(CHEMBL2283221)
Affinity DataIC50: 240nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488130(CHEMBL2283208)
Affinity DataIC50: 280nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488116(CHEMBL2283209)
Affinity DataIC50: 300nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488136(CHEMBL2283222)
Affinity DataIC50: 320nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488123(CHEMBL2283223)
Affinity DataIC50: 370nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488122(CHEMBL2283224)
Affinity DataIC50: 460nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488119(CHEMBL2283210)
Affinity DataIC50: 560nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488120(CHEMBL2283225)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488121(CHEMBL2283226)
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50255245(3-chloro-1-(4-hydroxyphenyl)propan-1-one | CHEMBL5...)
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of GABA transaminase in rat brain by Kitz-Wilson plotMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50488118(CHEMBL2283227)
Affinity DataIC50: 4.96E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177407(1-(4-hydroxyphenyl)prop-2-en-1-one | 4-acryloylphe...)
Affinity DataIC50: 5.48E+3nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50488135(CHEMBL2283228)
Affinity DataIC50: 6.54E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50561618(CHEMBL4746439)
Affinity DataIC50: 9.69E+3nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50488129(CHEMBL2283211)
Affinity DataIC50: 9.95E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488128(CHEMBL2283212)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632823(CHEMBL4740703)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Mouse)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50510591(CHEMBL4521189)
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177412(4-(aminomethyl)phenol | 4-hydroxybenzylamine | CHE...)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177410(4-hydroxy-3-nitrobenzaldehyde | CHEMBL378361)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50488138(CHEMBL2283213)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50177411(4-hydroxybenzaldehyde | 4-formylphenol | p-formylp...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of GABA transaminase in rat brain by Kitz-Wilson plotMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177411(4-hydroxybenzaldehyde | 4-formylphenol | p-formylp...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50488141(CHEMBL2283214)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177405(4-hydroxy-3-methoxybenzaldehyde | vanillin | 3-met...)
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632821(CHEMBL4750359)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632822(CHEMBL5408239)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
LigandPNGBDBM50488127(CHEMBL2283215)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488137(CHEMBL2283216)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488115(CHEMBL2283217)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488126(CHEMBL2283218)
Affinity DataIC50: 2.59E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

LigandPNGBDBM50488125(CHEMBL2283219)
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632820(CHEMBL5404015)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Mouse)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50118886(CHEMBL89598 | 4-Amino-hex-5-enoic acid | VIGABATRI...)
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50118886(CHEMBL89598 | 4-Amino-hex-5-enoic acid | VIGABATRI...)
Affinity DataIC50: 4.12E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50488124(CHEMBL2283220)
Affinity DataIC50: 4.41E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

Target4-aminobutyrate aminotransferase, mitochondrial(Mouse)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50510593(CHEMBL4569177)
Affinity DataIC50: 5.14E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Mouse)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50510592(CHEMBL4452708)
Affinity DataIC50: 5.81E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177402(1-(4-hydroxyphenyl)propan-1-one | Paroxypropione |...)
Affinity DataIC50: 1.76E+5nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177409(1-(4-hydroxyphenyl)ethanone | 4'-hydroxyacetopheno...)
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177403((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(4-(hydroxyme...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376755(CHEMBL535643)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50009001(CHEMBL8260 | Baicalein | 5,6,7-Trihydroxyflavone |...)
Affinity DataIC50: 1.28E+7nMAssay Description:Inhibition of GABA transaminase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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