Compile Data Set for Download or QSAR
Report error Found 23 of ic50 data for polymerid = 49000507,50000883
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50299218(Cpd66 | 8-(2-Methoxyphenyl)-1-methyl-7-(2'-methyl-...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of EphB1 by [gamma33-P]ATP based assayMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50244430(AP24149 | CHEMBL488840 | 9-(2,6-dimethylstyryl)-N-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of EphB1More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human EPHB1 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50577169(CHEMBL4846921)
Affinity DataIC50: 30nMAssay Description:Inhibition of EphB1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 60.3nMAssay Description:Inhibition of human EPHB1 using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 110nMAssay Description:Inhibition of EPHB1More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 128nMAssay Description:Inhibition of EPHB1 (unknown origin) incubated for 1 hr by spectrophotometric analysisMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50563891(CHEMBL4793380)
Affinity DataIC50: 388nMAssay Description:Inhibition of recombinant human EphB1 (564 to end residues) using KVEKIGEGTYGVVYK as substrate incubated for 40 mins in presence of [gamma-33ATP] by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50618607(CHEMBL5425418)
Affinity DataIC50: 632nMAssay Description:Inhibition of full length NanoLuc fused EPHB1 (unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo substrate incubated for 2 hrs in p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50358591(CHEMBL1923983)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of EphB1More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 3.04E+3nMAssay Description:Inhibition of EPHB1-mediated proliferation of mouse BAF3 cells transformed with TEL-Kinase constructMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50428059(CHEMBL2322989)
Affinity DataIC50: 3.80E+3nMAssay Description:Displacement of ephrin-B1-Fc from EphB1 receptor Fc ectodomain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50357884(CHEMBL1916359)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human EphB1More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50429867(CHEMBL2333365)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EPHB1 (unknown origin)More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50509949(CHEMBL4475216 | US11667631, Example 29)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EphB1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human EphB1 (564 to end residues) using KVEKIGEGTYGVV as substrate after 40 mins in presence of [gamma-33ATP] by radiometri...More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human EPHB1 using poly[Glu:Tyr] (4:1) as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50389320(CHEMBL2063926)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EPHB1 by FRET assayMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50359359(CHEMBL1929238)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of EPHB1More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50182493(CHEMBL3818247 | US9512121, 22)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of EPHB1 (unknown origin) incubated for 1 hr by spectrophotometric analysisMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50551201(CHEMBL4761556)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of biotinylated ephrin-B1-Fc from rat EphB1 Fc preincubated for 1 hr followed by ephrin-B1-FC addition and measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)
Affinity DataIC50: 3.77E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPHB1 catalytic domain expressed in baculovirus expression system using tyrosine-2 peptide as substrate in...More data for this Ligand-Target Pair
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PubMed
TargetEphrin type-B receptor 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50380246(CHEMBL2017214)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of EPHB1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed